Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 6008
TargetDiscoidin domain-containing receptor 2(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM50237710(AMN 107 | AMN107 | 4-methyl-N-[3-(4-methyl-1H-imid...)
Affinity DataIC50: 0.5nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104010(DDR1-IN-2)
Affinity DataEC50:  9nMAssay Description:The enzyme kinase assay was carried out using the Lanthascreen technology.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM50237710(AMN 107 | AMN107 | 4-methyl-N-[3-(4-methyl-1H-imid...)
Affinity DataIC50: 43nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104010(DDR1-IN-2)
Affinity DataIC50: 47.6nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104009(DDR1-IN-1)
Affinity DataEC50:  86nMAssay Description:The enzyme kinase assay was carried out using the Lanthascreen technology.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104009(DDR1-IN-1)
Affinity DataIC50: 105nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDiscoidin domain-containing receptor 2(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104010(DDR1-IN-2)
Affinity DataIC50: 145nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 337nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM104009(DDR1-IN-1)
Affinity DataIC50: 413nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Massachusetts General Hospital and Harvard Medical School

LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 675nMAssay Description:Tet inducible human DDR1 over-expressing U2OS was pre-treated by media containing each of the compound for 1 hour and treated by changing the media t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed