Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50044801
TargetCathepsin S(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030823(CHEMBL3342553)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mouse cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030822(CHEMBL3342554)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of mouse cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030823(CHEMBL3342553)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of human cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCathepsin S(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030822(CHEMBL3342554)
Affinity DataIC50: 12nMAssay Description:Inhibition of human cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030816(CHEMBL3342550)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030817(CHEMBL3342551)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030816(CHEMBL3342550)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of mouse cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030817(CHEMBL3342551)
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of mouse cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030821(CHEMBL3342552)
Affinity DataIC50: 3.93E+3nMAssay Description:Inhibition of mouse cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetCathepsin S(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030821(CHEMBL3342552)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human cathepsin S using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50030816(CHEMBL3342550)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human cathepsin L using benzyloxycarbonyl-L-Leucyl-L-Arginine 4-Methyl-coumaryl-7-amide substrate by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed