Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50046012
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50091030(CHEMBL3582033)
Affinity DataIC50: 10nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50317323(N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-4-yl)thieno...)
Affinity DataIC50: 12nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090969(CHEMBL3582034)
Affinity DataIC50: 13nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50317324(N-(4-(6,7-dimethoxyquinolin-4-yloxy)-3-fluoropheny...)
Affinity DataIC50: 16nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090968(CHEMBL3582035)
Affinity DataIC50: 17nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50317323(N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-4-yl)thieno...)
Affinity DataIC50: 30nMAssay Description:Inhibition of RON phosphorylation in human PC3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50317323(N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-4-yl)thieno...)
Affinity DataIC50: 30nMAssay Description:Inhibition of RON phosphorylation in human HT29 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090966(CHEMBL3582037)
Affinity DataIC50: 44nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090967(CHEMBL3582036)
Affinity DataIC50: 95nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50091026(CHEMBL3580678)
Affinity DataIC50: 580nMAssay Description:Inhibition of RON (unknown origin) transfected in 293T cells assessed as autophosporylated level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090968(CHEMBL3582035)
Affinity DataIC50: 670nMAssay Description:Inhibition of phosphorylation of c-Met in human MKN45 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50317324(N-(4-(6,7-dimethoxyquinolin-4-yloxy)-3-fluoropheny...)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of phosphorylation of c-Met in human MKN45 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090969(CHEMBL3582034)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of phosphorylation of c-Met in human MKN45 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090967(CHEMBL3582036)
Affinity DataIC50: 3.77E+3nMAssay Description:Inhibition of phosphorylation of c-Met in human MKN45 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50090966(CHEMBL3582037)
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of phosphorylation of c-Met in human MKN45 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Chemrf Laboratories

Curated by ChEMBL
LigandPNGBDBM50317323(N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-4-yl)thieno...)
Affinity DataIC50: 6.87E+3nMAssay Description:Inhibition of phosphorylation of c-Met in human MKN45 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2016
Entry Details Article
PubMed