TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 0.990nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 114nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 171nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 865nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 991nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 1.13E+3nMAssay Description:Displacement of [3H]DAMGO from rat cortical MOR by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 1.28E+3nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 2.27E+3nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 3.23E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 3.32E+3nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 4.45E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 5.07E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 5.33E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 8.16E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 8.43E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 8.53E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]DPDPE from rat cortical DOR after 2.5 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U69,593 from guinea pig KOR after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 678nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:Agonist activity at human MOR expressed in CHO cells assessed as induction of membrane potential change measured every 3 secs for 30 secs by fluoresc...More data for this Ligand-Target Pair