Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50048149
TargetTransthyretin(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50206384(CHEMBL3917629)
Affinity DataIC50:  1.49E+3nMAssay Description:Inhibition of wild type TTR (unknown origin) assessed as inhibition of acid-mediated amyloidogenesis by measuring fibril formation preincubated with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50197883(CHEBI:78538 | FX-1006 | Tafamidis | US10377729, Co...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of wild type TTR (unknown origin) assessed as inhibition of acid-mediated amyloidogenesis by measuring fibril formation preincubated with ...More data for this Ligand-Target Pair
TargetTransthyretin(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50206387(CHEMBL3898378)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of wild type TTR (unknown origin) assessed as inhibition of acid-mediated amyloidogenesis by measuring fibril formation preincubated with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50206385(CHEMBL3976323)
Affinity DataIC50:  2.06E+3nMAssay Description:Inhibition of wild type TTR (unknown origin) assessed as inhibition of acid-mediated amyloidogenesis by measuring fibril formation preincubated with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50206388(CHEMBL3899454)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibition of wild type TTR (unknown origin) assessed as inhibition of acid-mediated amyloidogenesis by measuring fibril formation preincubated with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransthyretin(Homo sapiens (Human))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50206386(CHEMBL3987064)
Affinity DataIC50:  2.59E+3nMAssay Description:Inhibition of wild type TTR (unknown origin) assessed as inhibition of acid-mediated amyloidogenesis by measuring fibril formation preincubated with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed