Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50048071
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203462BDBM50203462(CHEMBL3931161)
Affinity DataIC50: 31nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203462BDBM50203462(CHEMBL3931161)
Affinity DataIC50: 40nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL-17A release after 4 days by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203506BDBM50203506(CHEMBL3977048)
Affinity DataIC50: 44nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203497BDBM50203497(CHEMBL3924898)
Affinity DataIC50: 54nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203542BDBM50203542(CHEMBL3218921)
Affinity DataIC50: 60nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50445877BDBM50445877(CHEMBL3105681)
Affinity DataIC50: 80nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203513BDBM50203513(CHEMBL3913238)
Affinity DataIC50: 88nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203493BDBM50203493(CHEMBL3912204)
Affinity DataIC50: 120nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203508BDBM50203508(CHEMBL3968165)
Affinity DataIC50: 140nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203493BDBM50203493(CHEMBL3912204)
Affinity DataIC50: 150nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL-17A release after 4 days by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203541BDBM50203541(CHEMBL3948265)
Affinity DataIC50: 240nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203459BDBM50203459(CHEMBL3894222)
Affinity DataIC50: 260nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203496BDBM50203496(CHEMBL3929577)
Affinity DataIC50: 300nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203465BDBM50203465(CHEMBL3929358)
Affinity DataIC50: 310nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203546BDBM50203546(CHEMBL3920663)
Affinity DataIC50: 370nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203487BDBM50203487(CHEMBL3961289)
Affinity DataIC50: 590nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203463BDBM50203463(CHEMBL3979349)
Affinity DataIC50: 720nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203459BDBM50203459(CHEMBL3894222)
Affinity DataIC50: 800nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203544BDBM50203544(CHEMBL3928131)
Affinity DataIC50: 820nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203516BDBM50203516(CHEMBL3967961)
Affinity DataIC50: 1.10E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203544BDBM50203544(CHEMBL3928131)
Affinity DataIC50: 1.10E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203490BDBM50203490(CHEMBL3905660)
Affinity DataIC50: 1.20E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203504BDBM50203504(CHEMBL3938404)
Affinity DataIC50: 1.20E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203542BDBM50203542(CHEMBL3218921)
Affinity DataIC50: 1.30E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203508BDBM50203508(CHEMBL3968165)
Affinity DataIC50: 1.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203514BDBM50203514(CHEMBL3977144)
Affinity DataIC50: 1.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203488BDBM50203488(CHEMBL3957141)
Affinity DataIC50: 1.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203516BDBM50203516(CHEMBL3967961)
Affinity DataIC50: 1.90E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203460BDBM50203460(CHEMBL3956929)
Affinity DataIC50: 2.10E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203520BDBM50203520(CHEMBL3943864)
Affinity DataIC50: 2.50E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203518BDBM50203518(CHEMBL3942787)
Affinity DataIC50: 2.50E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203523BDBM50203523(CHEMBL3933686)
Affinity DataIC50: 2.60E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203543BDBM50203543(CHEMBL3951385)
Affinity DataIC50: 2.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203511BDBM50203511(CHEMBL3911834)
Affinity DataIC50: 2.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203509BDBM50203509(CHEMBL3948459)
Affinity DataIC50: 3.50E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203515BDBM50203515(CHEMBL3920454)
Affinity DataIC50: 3.60E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203507BDBM50203507(CHEMBL3915908)
Affinity DataIC50: 3.60E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203504BDBM50203504(CHEMBL3938404)
Affinity DataIC50: 3.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203462BDBM50203462(CHEMBL3931161)
Affinity DataKd:  4.00E+3nMAssay Description:Activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203490BDBM50203490(CHEMBL3905660)
Affinity DataIC50: 4.10E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203539BDBM50203539(CHEMBL3950318)
Affinity DataIC50: 4.20E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203522BDBM50203522(CHEMBL3914641)
Affinity DataIC50: 4.30E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203518BDBM50203518(CHEMBL3942787)
Affinity DataIC50: 4.40E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203499BDBM50203499(CHEMBL3947885)
Affinity DataIC50: 4.50E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203500BDBM50203500(CHEMBL3986751)
Affinity DataIC50: 4.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203505BDBM50203505(CHEMBL3976477)
Affinity DataIC50: 4.80E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203510BDBM50203510(CHEMBL3939711)
Affinity DataIC50: 5.00E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203517BDBM50203517(CHEMBL3933815)
Affinity DataIC50: 5.60E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203503BDBM50203503(CHEMBL3982499)
Affinity DataIC50: 5.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RARgamma LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Galderma R & D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50203521BDBM50203521(CHEMBL3938989)
Affinity DataIC50: 5.90E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2018
Entry Details Article
PubMed
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