Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50049156
TargetCyclin-dependent kinase 2(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235359BDBM50235359(CHEMBL4088242)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235343BDBM50235343(CHEMBL4103249)
Affinity DataIC50: 1nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235335BDBM50235335(CHEMBL4092981)
Affinity DataIC50: 2nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235348BDBM50235348(CHEMBL4078988)
Affinity DataIC50: 3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235342BDBM50235342(NU-6102 | CHEMBL319467)
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235346BDBM50235346(CHEMBL4102518)
Affinity DataIC50: 8nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235347BDBM50235347(CHEMBL4078246)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235349BDBM50235349(CHEMBL4065402)
Affinity DataIC50: 17nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235336BDBM50235336(CHEMBL4085238)
Affinity DataIC50: 18nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235354BDBM50235354(CHEMBL4069161)
Affinity DataIC50: 19nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235344BDBM50235344(CHEMBL4086832)
Affinity DataIC50: 19nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235345BDBM50235345(CHEMBL4105278)
Affinity DataIC50: 24nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235337BDBM50235337(CHEMBL4062554)
Affinity DataIC50: 26nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235340BDBM50235340(CHEMBL4101626)
Affinity DataIC50: 26nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235355BDBM50235355(CHEMBL4081027)
Affinity DataIC50: 39nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235334BDBM50235334(CHEMBL4070391)
Affinity DataIC50: 44nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235356BDBM50235356(CHEMBL4097571)
Affinity DataIC50: 52nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235343BDBM50235343(CHEMBL4103249)
Affinity DataIC50: 97nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235353BDBM50235353(CHEMBL4090226)
Affinity DataIC50: 220nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235342BDBM50235342(NU-6102 | CHEMBL319467)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235332BDBM50235332(CHEMBL4094205)
Affinity DataIC50: 290nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235342BDBM50235342(NU-6102 | CHEMBL319467)
Affinity DataIC50: 480nMAssay Description:Inhibition of human CDK5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235345BDBM50235345(CHEMBL4105278)
Affinity DataIC50: 570nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235343BDBM50235343(CHEMBL4103249)
Affinity DataIC50: 570nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235357BDBM50235357(CHEMBL4089837)
Affinity DataIC50: 580nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235345BDBM50235345(CHEMBL4105278)
Affinity DataIC50: 730nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235335BDBM50235335(CHEMBL4092981)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235335BDBM50235335(CHEMBL4092981)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235361BDBM50235361(CHEMBL4074015)
Affinity DataIC50: 830nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235344BDBM50235344(CHEMBL4086832)
Affinity DataIC50: 940nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5530BDBM5530(6-(cyclohexylmethoxy)-N-phenyl-9H-purin-2-amine | ...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235337BDBM50235337(CHEMBL4062554)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235342BDBM50235342(NU-6102 | CHEMBL319467)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235329BDBM50235329(CHEMBL4061761)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235339BDBM50235339(CHEMBL4073211)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235336BDBM50235336(CHEMBL4085238)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235337BDBM50235337(CHEMBL4062554)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human CDK1/Cyclin B expressed in baculovirus infected Sf9 cells using PKTPKKAKKL-NH2 as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235343BDBM50235343(CHEMBL4103249)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235335BDBM50235335(CHEMBL4092981)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human CDK5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235337BDBM50235337(CHEMBL4062554)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235342BDBM50235342(NU-6102 | CHEMBL319467)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235337BDBM50235337(CHEMBL4062554)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human CDK5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235336BDBM50235336(CHEMBL4085238)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk9/human full-length Cyclin T expressed in baculovirus infected Sf21 insect cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235336BDBM50235336(CHEMBL4085238)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human CDK5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235351BDBM50235351(CHEMBL4102300)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235330BDBM50235330(CHEMBL4081980)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235345BDBM50235345(CHEMBL4105278)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235335BDBM50235335(CHEMBL4092981)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235336BDBM50235336(CHEMBL4085238)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of recombinant human full-length C-terminal His6-tagged Cdk7/recombinant human full-length Cyclin H expressed in baculovirus infected Sf21...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
TargetCyclin-A2(Bovine)
Newcastle University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235352BDBM50235352(CHEMBL4084337)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human GST-tagged CDK2/bovine His-tagged Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2019
Entry Details Article
PubMed
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