Affinity DataKi: 158nMAssay Description:Displacement of [3H]NMS from wild-type human mAChR2 expressed in Flp-in-CHO cell membranes in presence of mAChR2 agonist xanomeline after 90 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 3.16E+3nMAssay Description:Displacement of [3H]NMS from wild-type human mAChR2 expressed in Flp-In-CHO cell membranes in presence of mAChR2 agonist acetylcholine after 90 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant full length BTK (unknown origin) using peptide substrate by capillary elctrophoresisMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1(Homo sapiens (Human))
Intellisyn Pharma
Curated by ChEMBL
Intellisyn Pharma
Curated by ChEMBL
Affinity DataEC50: 79nMAssay Description:Positive allosteric modulation at human GABA-B 1b expressed in CHO cells co-expressing rat GABA-B2 assessed as potentiation of GABA-induced inhibitio...More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+4nMAssay Description:Positive allosteric modulatory activity at recombinant human glycine alpha1 receptor expressed in HEK293 cells assessed as potentiation of glycine-in...More data for this Ligand-Target Pair