Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity to human serum albumin by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity to human serum albumin assessed as inhibition constant by NMR spectroscopyMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+5nMAssay Description:Binding affinity to factor D (unknown origin) by 19F-NMR spectroscopyMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+5nMAssay Description:Binding affinity to factor D (unknown origin) by 19F-NMR spectroscopyMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of recombinant human factor D expressed in Escherichia coli using Z-Lys-thiobenzyl as substrate after 1 hr by spectrofluorimetryMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Escherichia coli PPAT after 5 mins by reverse ATP-generating-luciferase assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+5nMAssay Description:Binding affinity to Nurr1 (unknown origin) by 1H-STD-NMR spectroscopyMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+6nMAssay Description:Binding affinity to human DC-SIGN ECD expressed in Escherichia coli BL21(DE3) after 1 hr by Man-Fl-BSA assayMore data for this Ligand-Target Pair
Affinity DataKd: 4.10E+4nMAssay Description:Binding affinity to human serum albumin by ITCMore data for this Ligand-Target Pair
Affinity DataKd: 2.10E+6nMAssay Description:Binding affinity to human DC-SIGN ECD expressed in Escherichia coli BL21(DE3) after 1 hr by Man-Fl-BSA assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to Nurr1 (unknown origin) by 1H-STD-NMR spectroscopyMore data for this Ligand-Target Pair
TargetBifunctional UDP-N-acetylglucosamine 2-epimerase/N-acetylmannosamine kinase(Homo sapiens)
Lavis
Curated by ChEMBL
Lavis
Curated by ChEMBL
Affinity DataKd: 8.00E+4nMAssay Description:Binding affinity to His-tagged human MNK expressed in Escherichia coli BL21(DE3) in presence of ATP by 9F-NMR spectroscopy analysisMore data for this Ligand-Target Pair
TargetBifunctional UDP-N-acetylglucosamine 2-epimerase/N-acetylmannosamine kinase(Homo sapiens)
Lavis
Curated by ChEMBL
Lavis
Curated by ChEMBL
Affinity DataKd: 9.00E+5nMAssay Description:Binding affinity to His-tagged human MNK expressed in Escherichia coli BL21(DE3) in presence of ATP by 9F-NMR spectroscopy analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to human DC-SIGN ECD expressed in Escherichia coli BL21(DE3) after 1 hr by Man-Fl-BSA assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.60E+6nMAssay Description:Binding affinity to human DC-SIGN ECD expressed in Escherichia coli BL21(DE3) after 1 hr by Man-Fl-BSA assayMore data for this Ligand-Target Pair
Affinity DataKd: 4.18E+4nMAssay Description:Binding affinity to human serum albumin by NMR spectroscopyMore data for this Ligand-Target Pair