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Found 6 Enz. Inhib. hit(s) with all data for entry = 50009540
TargetTubulin beta chain(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529724(CHEMBL4437037)
Affinity DataIC50:  2.09E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization preincubated for 30 mins and measured every 2 mins for 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529724(CHEMBL4437037)
Affinity DataIC50:  2.09E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization preincubated for 30 mins and measured every 2 mins for 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization preincubated for 30 mins and measured every 2 mins for 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization preincubated for 30 mins and measured every 2 mins for 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529723(CHEMBL4474171)
Affinity DataIC50:  2.54E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization preincubated for 30 mins and measured every 2 mins for 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529723(CHEMBL4474171)
Affinity DataIC50:  2.54E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization preincubated for 30 mins and measured every 2 mins for 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed