Compile Data Set for Download or QSAR
Report error Found 257 Enz. Inhib. hit(s) with all data for entry = 50007858
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513361(CHEMBL4567766)
Affinity DataKi:  1nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataKi:  1nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataKi:  2nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513360(CHEMBL4573390)
Affinity DataKi:  2nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50151923(CHEMBL3774537)
Affinity DataKi:  2nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50151923(CHEMBL3774537)
Affinity DataKi:  3nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513344(CHEMBL4447515)
Affinity DataKi:  3nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513361(CHEMBL4567766)
Affinity DataKi:  3nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513348(CHEMBL4585876)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 4nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513348(CHEMBL4585876)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513344(CHEMBL4447515)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 5nMAssay Description:Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 5nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513360(CHEMBL4573390)
Affinity DataKi:  5nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 6nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 6nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 7nMAssay Description:Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataKi:  7nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 9nMAssay Description:Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 11nMAssay Description:Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513348(CHEMBL4585876)
Affinity DataIC50: 12nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513372(CHEMBL4440395)
Affinity DataIC50: 12nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513352(CHEMBL4592908)
Affinity DataIC50: 12nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 13nMAssay Description:Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513360(CHEMBL4573390)
Affinity DataIC50: 14nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5C(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 14nMAssay Description:Inhibition of KDM5C (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 15nMAssay Description:Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513372(CHEMBL4440395)
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 16nMAssay Description:Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513346(CHEMBL4525269)
Affinity DataKi:  16nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513351(CHEMBL4516101)
Affinity DataIC50: 17nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513361(CHEMBL4567766)
Affinity DataIC50: 17nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 17nMAssay Description:Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513374(CHEMBL4466130)
Affinity DataIC50: 18nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513352(CHEMBL4592908)
Affinity DataIC50: 19nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513348(CHEMBL4585876)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513357(CHEMBL4590283)
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513354(CHEMBL4558689)
Affinity DataIC50: 21nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataIC50: 21nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 22nMAssay Description:Inhibition of full length human KDM4B assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbiotin) as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 4A(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 22nMAssay Description:Inhibition of full length human KDM4A A482E mutant assessed as decrease in demethylation of substrate using peptide (ARTKQTARK(Me3)STGGKAPRKQLA-GGKbi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataIC50: 23nMAssay Description:Inhibition of full length human KDM5B assessed as decrease in demethylation of substrate using peptide ARTK(me3)QTARKSTGGKAPRKQLA-GGK-biotin as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetLysine-specific demethylase 5B(Human)
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513373(CHEMBL4538741)
Affinity DataIC50: 23nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 257 total ) | Next | Last >>
Jump to: