Compile Data Set for Download or QSAR
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Found 35 Enz. Inhib. hit(s) with all data for entry = 50011773
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550973(CHEMBL4784857)
Affinity DataIC50:  40nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550969(CHEMBL4744389)
Affinity DataIC50:  44nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550967(CHEMBL4762199)
Affinity DataIC50:  47nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550977(CHEMBL4740282)
Affinity DataIC50:  59nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550975(CHEMBL4742337)
Affinity DataIC50:  76nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550976(CHEMBL4799779)
Affinity DataIC50:  83nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550970(CHEMBL4750433)
Affinity DataIC50:  120nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550968(CHEMBL4743350)
Affinity DataIC50:  190nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550971(CHEMBL4783756)
Affinity DataIC50:  190nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550966(CHEMBL4761281)
Affinity DataIC50:  230nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550972(CHEMBL4796411)
Affinity DataIC50:  270nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550983(CHEMBL4749117)
Affinity DataIC50:  350nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550974(CHEMBL4795875)
Affinity DataIC50:  360nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550982(CHEMBL4764779)
Affinity DataIC50:  430nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550981(CHEMBL4776485)
Affinity DataIC50:  590nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550980(CHEMBL4745258)
Affinity DataIC50:  610nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550979(CHEMBL4785060)
Affinity DataIC50:  660nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550978(CHEMBL4782382)
Affinity DataIC50:  680nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550984(CHEMBL4751384)
Affinity DataIC50:  740nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-p-nitroanilide as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550973(CHEMBL4784857)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human ERG expressed in CHO cells by manual patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50244791((2-Fluoro-4-methanesulfonyl-phenyl)-{6-[4-(3-isopr...)
Affinity DataEC50:  640nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550979(CHEMBL4785060)
Affinity DataEC50:  2.56E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550980(CHEMBL4745258)
Affinity DataEC50:  3.99E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550981(CHEMBL4776485)
Affinity DataEC50:  1.85E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550982(CHEMBL4764779)
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550983(CHEMBL4749117)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550984(CHEMBL4751384)
Affinity DataEC50:  4.02E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550978(CHEMBL4782382)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550977(CHEMBL4740282)
Affinity DataEC50:  650nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550973(CHEMBL4784857)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550970(CHEMBL4750433)
Affinity DataEC50:  830nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550969(CHEMBL4744389)
Affinity DataEC50:  600nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550968(CHEMBL4743350)
Affinity DataEC50:  3.13E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Chinese Academy Of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550974(CHEMBL4795875)
Affinity DataEC50:  1.93E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed