Affinity DataKi: 30nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of His/GST-tagged PKN2 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.19E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.69E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.85E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.11E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.19E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.29E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.91E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.94E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.11E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.24E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.38E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.59E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.02E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.88E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.37E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.77E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))
University Of Sussex
Curated by ChEMBL
University Of Sussex
Curated by ChEMBL
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged CLK4 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.12E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.45E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.02E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.71E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.06E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.59E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.13E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.85E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.88E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair