Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 50011123
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  30nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  40nMAssay Description:Inhibition of His/GST-tagged PKN2 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545113(CHEMBL4647033)
Affinity DataKi:  80nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  540nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545105(CHEMBL4635777)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545108(CHEMBL4646744)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545113(CHEMBL4647033)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545111(CHEMBL4634210)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545101(CHEMBL4636367)
Affinity DataKi:  2.69E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM55759(2-(4-pyridyl)-1H-benzimidazole | 2-pyridin-4-yl-1H...)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545105(CHEMBL4635777)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545104(CHEMBL4645636)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545107(CHEMBL4637286)
Affinity DataKi:  8.11E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545102(CHEMBL185288)
Affinity DataKi:  8.19E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545112(CHEMBL160012)
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545109(CHEMBL4632420)
Affinity DataKi:  1.56E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545111(CHEMBL4634210)
Affinity DataKi:  1.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545109(CHEMBL4632420)
Affinity DataKi:  1.91E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545106(CHEMBL4649365)
Affinity DataKi:  1.94E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545110(CHEMBL4638916)
Affinity DataKi:  2.11E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM55759(2-(4-pyridyl)-1H-benzimidazole | 2-pyridin-4-yl-1H...)
Affinity DataKi:  2.24E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545103(CHEMBL4640475)
Affinity DataKi:  2.38E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545101(CHEMBL4636367)
Affinity DataKi:  2.59E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545106(CHEMBL4649365)
Affinity DataKi:  2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545110(CHEMBL4638916)
Affinity DataKi:  2.78E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545108(CHEMBL4646744)
Affinity DataKi:  2.89E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545104(CHEMBL4645636)
Affinity DataKi:  3.02E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545102(CHEMBL185288)
Affinity DataKi:  3.25E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545107(CHEMBL4637286)
Affinity DataKi:  4.88E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545112(CHEMBL160012)
Affinity DataKi:  5.37E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545103(CHEMBL4640475)
Affinity DataKi:  6.77E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged CLK4 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataIC50:  64nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545113(CHEMBL4647033)
Affinity DataIC50:  170nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545105(CHEMBL4635777)
Affinity DataIC50:  2.12E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545108(CHEMBL4646744)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545113(CHEMBL4647033)
Affinity DataIC50:  4.45E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545111(CHEMBL4634210)
Affinity DataIC50:  5.02E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545101(CHEMBL4636367)
Affinity DataIC50:  5.40E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM55759(2-(4-pyridyl)-1H-benzimidazole | 2-pyridin-4-yl-1H...)
Affinity DataIC50:  7.71E+3nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545105(CHEMBL4635777)
Affinity DataIC50:  1.06E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545104(CHEMBL4645636)
Affinity DataIC50:  1.38E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545107(CHEMBL4637286)
Affinity DataIC50:  1.62E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545102(CHEMBL185288)
Affinity DataIC50:  1.64E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545112(CHEMBL160012)
Affinity DataIC50:  2.59E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545109(CHEMBL4632420)
Affinity DataIC50:  3.13E+4nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545111(CHEMBL4634210)
Affinity DataIC50:  3.85E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545109(CHEMBL4632420)
Affinity DataIC50:  3.88E+4nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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