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Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50016231
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593405(CHEMBL5178783)
Affinity DataEC50:  33nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593381(CHEMBL5192713)
Affinity DataEC50:  64nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593406(CHEMBL5206362)
Affinity DataEC50:  88nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593403(CHEMBL5199523)
Affinity DataEC50:  91nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593378(CHEMBL5202704)
Affinity DataEC50:  132nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593401(CHEMBL5192503)
Affinity DataEC50:  133nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593373(CHEMBL5182581)
Affinity DataEC50:  137nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593405(CHEMBL5178783)
Affinity DataEC50:  145nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593387(CHEMBL5187664)
Affinity DataEC50:  146nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593377(CHEMBL5186323)
Affinity DataEC50:  150nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593371(CHEMBL5189637)
Affinity DataEC50:  165nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593394(CHEMBL5209446)
Affinity DataEC50:  187nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593381(CHEMBL5192713)
Affinity DataEC50:  229nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593376(CHEMBL5180586)
Affinity DataEC50:  239nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593378(CHEMBL5202704)
Affinity DataEC50:  335nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593394(CHEMBL5209446)
Affinity DataEC50:  360nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593406(CHEMBL5206362)
Affinity DataEC50:  371nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593403(CHEMBL5199523)
Affinity DataEC50:  430nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593379(CHEMBL5198649)
Affinity DataEC50:  448nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593388(CHEMBL5183734)
Affinity DataEC50:  484nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593382(CHEMBL5195437)
Affinity DataEC50:  493nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593377(CHEMBL5186323)
Affinity DataEC50:  563nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593402(CHEMBL5194469)
Affinity DataEC50:  577nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593392(CHEMBL5190916)
Affinity DataEC50:  592nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593376(CHEMBL5180586)
Affinity DataEC50:  601nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593401(CHEMBL5192503)
Affinity DataEC50:  607nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593397(CHEMBL1419647)
Affinity DataEC50:  609nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593404(CHEMBL5209389)
Affinity DataEC50: >677nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593373(CHEMBL5182581)
Affinity DataEC50:  702nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593371(CHEMBL5189637)
Affinity DataEC50:  720nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593400(CHEMBL5185425)
Affinity DataEC50:  723nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593387(CHEMBL5187664)
Affinity DataEC50:  730nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593398(CHEMBL5186610)
Affinity DataEC50:  782nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593374(CHEMBL5205455)
Affinity DataEC50:  962nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593402(CHEMBL5194469)
Affinity DataEC50:  1.17E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593382(CHEMBL5195437)
Affinity DataEC50:  1.28E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593388(CHEMBL5183734)
Affinity DataEC50:  1.29E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593395(CHEMBL5185110)
Affinity DataEC50:  1.40E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593380(CHEMBL5178207)
Affinity DataEC50:  1.45E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593379(CHEMBL5198649)
Affinity DataEC50:  1.54E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593386(CHEMBL5207050)
Affinity DataEC50:  1.74E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593400(CHEMBL5185425)
Affinity DataEC50:  2.87E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593393(CHEMBL5170104)
Affinity DataEC50:  2.96E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593392(CHEMBL5190916)
Affinity DataEC50: >3.00E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593374(CHEMBL5205455)
Affinity DataEC50:  3.13E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593391(CHEMBL5200886)
Affinity DataEC50:  3.47E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593393(CHEMBL5170104)
Affinity DataEC50:  3.84E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593380(CHEMBL5178207)
Affinity DataEC50:  3.92E+3nMAssay Description:Activation of GIRK1/4 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593399(CHEMBL5199370)
Affinity DataEC50: >4.00E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska

Curated by ChEMBL
LigandPNGBDBM50593389(CHEMBL5178976)
Affinity DataEC50:  4.20E+3nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
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