Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50015139
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583213BDBM50583213(CHEMBL5086997)
Affinity DataEC50:  91nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells assessed as increase in calcium response at -90 mV holding potential measured at 1 to 2 days by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583211BDBM50583211(CHEMBL5078247)
Affinity DataEC50:  110nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells assessed as increase in calcium response at -90 mV holding potential measured at 1 to 2 days by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Human)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583211BDBM50583211(CHEMBL5078247)
Affinity DataEC50:  190nMAssay Description:Potentiation of human KCa2.3 expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiology relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Human)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583213BDBM50583213(CHEMBL5086997)
Affinity DataEC50:  600nMAssay Description:Potentiation of human KCa2.3 expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583213BDBM50583213(CHEMBL5086997)
Affinity DataEC50:  640nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583211BDBM50583211(CHEMBL5078247)
Affinity DataEC50:  990nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583210BDBM50583210(CHEMBL5074700)
Affinity DataEC50:  1.89E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583212BDBM50583212(CHEMBL5076878)
Affinity DataEC50:  1.99E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583214BDBM50583214(CHEMBL5076032)
Affinity DataEC50:  2.97E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583216BDBM50583216(CHEMBL5081906)
Affinity DataEC50:  3.27E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583215BDBM50583215(CHEMBL5075016)
Affinity DataEC50:  3.45E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583223BDBM50583223(CHEMBL5077913)
Affinity DataEC50:  3.59E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583231BDBM50583231(CHEMBL5094656)
Affinity DataEC50:  4.32E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583220BDBM50583220(CHEMBL5079766)
Affinity DataEC50:  4.51E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583209BDBM50583209(CHEMBL5082158)
Affinity DataEC50:  5.03E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583219BDBM50583219(CHEMBL5088936)
Affinity DataEC50:  6.59E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275157BDBM50275157(N-cyclohexyl-2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-me...)
Affinity DataEC50:  7.48E+3nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583222BDBM50583222(CHEMBL5094693)
Affinity DataEC50:  1.38E+4nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583218BDBM50583218(CHEMBL5090801)
Affinity DataEC50: >3.00E+4nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583221BDBM50583221(CHEMBL5088498)
Affinity DataEC50:  3.88E+4nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583199BDBM50583199(CHEMBL5074647)
Affinity DataEC50:  4.97E+4nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583202BDBM50583202(CHEMBL5083279)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583203BDBM50583203(CHEMBL5081876)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583204BDBM50583204(CHEMBL5075501)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583205BDBM50583205(CHEMBL5069418)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583206BDBM50583206(CHEMBL5079218)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583207BDBM50583207(CHEMBL5088689)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583208BDBM50583208(CHEMBL5089976)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583217BDBM50583217(CHEMBL5084258)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583224BDBM50583224(CHEMBL5090420)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583225BDBM50583225(CHEMBL5076140)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583226BDBM50583226(CHEMBL5086120)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583196BDBM50583196(CHEMBL5084004)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583227BDBM50583227(CHEMBL5079837)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583197BDBM50583197(CHEMBL5079951)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583228BDBM50583228(CHEMBL5072517)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583198BDBM50583198(CHEMBL5090455)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583229BDBM50583229(CHEMBL5088379)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583230BDBM50583230(CHEMBL5075803)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583200BDBM50583200(CHEMBL5093708)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 2(Rat)
Chapman University School of Pharmacy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50583201BDBM50583201(CHEMBL5080805)
Affinity DataEC50: >1.00E+5nMAssay Description:Potentiation of rat KCa2.2a expressed in HEK293 cells at -90 mV holding potential measured at 1 to 2 days by patch clamp electrophysiologyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed