Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50016794
TargetGastric inhibitory polypeptide receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597204(CHEMBL5196841)
Affinity DataEC50:  12nMAssay Description:Positive allosteric modulator activity at human GIPR expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597206(CHEMBL5180960)
Affinity DataEC50:  16nMAssay Description:Positive allosteric modulator activity at human GLP-1R expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50597205(CHEMBL5184469)
Affinity DataEC50:  38nMAssay Description:Positive allosteric modulator activity at human GIPR expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed