Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50000297
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245586BDBM50245586(CHEMBL4077123)
Affinity DataEC50:  4.70nMAssay Description:Irreversible inhibition of recombinant full length wild-type 3'-FLAG-tagged BTK (unknown origin) expressed in HEK293T cells assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50357312BDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataKi:  4.80nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245588BDBM50245588(CHEMBL4085868)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245603BDBM50245603(CHEMBL4096207)
Affinity DataKi:  6nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245586BDBM50245586(CHEMBL4077123)
Affinity DataIC50: 7nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50357312BDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 8nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245586BDBM50245586(CHEMBL4077123)
Affinity DataKi:  8.90nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50161162BDBM50161162(AVL-292 | CC-292 | Spebrutinib | US9987276, Compou...)
Affinity DataIC50: 9nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403056BDBM50403056(CHEMBL2216827 | US9987276, Compound I-342 | US1059...)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50357312BDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245587BDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)
Affinity DataIC50: 12nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245587BDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)
Affinity DataKi:  14nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245603BDBM50245603(CHEMBL4096207)
Affinity DataIC50: 17nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245613BDBM50245613(CHEMBL4074840)
Affinity DataIC50: 19nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245602BDBM50245602(CHEMBL4088999)
Affinity DataIC50: 21nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245635BDBM50245635(CHEMBL4076543)
Affinity DataIC50: 21nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50161162BDBM50161162(AVL-292 | CC-292 | Spebrutinib | US9987276, Compou...)
Affinity DataKi:  21nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020471BDBM50020471(CHEMBL3290142)
Affinity DataIC50: 24nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020471BDBM50020471(CHEMBL3290142)
Affinity DataIC50: 25nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020471BDBM50020471(CHEMBL3290142)
Affinity DataKi:  27nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245586BDBM50245586(CHEMBL4077123)
Affinity DataEC50: <30nMAssay Description:Inhibition of BTK auto-phosphorylation at Y223 in human Pfeiffer cells measured after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245586BDBM50245586(CHEMBL4077123)
Affinity DataEC50: <30nMAssay Description:Inhibition of BTK auto-phosphorylation at Y223 in human U2932 cells measured after 4 hrs by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245642BDBM50245642(CHEMBL4059850)
Affinity DataIC50: 32nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245614BDBM50245614(CHEMBL4066223)
Affinity DataIC50: 34nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245612BDBM50245612(CHEMBL4101519)
Affinity DataIC50: 41nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245587BDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)
Affinity DataIC50: 54nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245617BDBM50245617(CHEMBL4067226)
Affinity DataIC50: 57nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245632BDBM50245632(CHEMBL4077618)
Affinity DataIC50: 63nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245646BDBM50245646(CHEMBL4066966)
Affinity DataIC50: 65nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245636BDBM50245636(CHEMBL4071818)
Affinity DataIC50: 68nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50020471BDBM50020471(CHEMBL3290142)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged wild-type EGFR (695 to end residues) expressed in baculovirus infected Sf9 insect cells using p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245628BDBM50245628(CHEMBL4064326)
Affinity DataIC50: 76nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245627BDBM50245627(CHEMBL4093610)
Affinity DataIC50: 86nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245639BDBM50245639(CHEMBL4088485)
Affinity DataIC50: 89nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245643BDBM50245643(CHEMBL4081428)
Affinity DataEC50: >100nMAssay Description:Irreversible inhibition of recombinant full length wild-type 3'-FLAG-tagged BTK (unknown origin) expressed in HEK293T cells assessed as reduction in ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245588BDBM50245588(CHEMBL4085868)
Affinity DataKi:  113nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245630BDBM50245630(CHEMBL4074645)
Affinity DataIC50: 114nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50357312BDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 123nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged wild-type EGFR (695 to end residues) expressed in baculovirus infected Sf9 insect cells using p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245604BDBM50245604(CHEMBL4076040)
Affinity DataIC50: 127nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50357312BDBM50357312(IBRUTINIB | US9181263, 1 | US9108973, Ref 1 | US92...)
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245643BDBM50245643(CHEMBL4081428)
Affinity DataIC50: 163nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245599BDBM50245599(CHEMBL4105457)
Affinity DataIC50: 187nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245637BDBM50245637(CHEMBL4093800)
Affinity DataIC50: 197nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403056BDBM50403056(CHEMBL2216827 | US9987276, Compound I-342 | US1059...)
Affinity DataKi:  209nMAssay Description:Reversible inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245629BDBM50245629(CHEMBL4081768)
Affinity DataIC50: 210nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245634BDBM50245634(CHEMBL4063526)
Affinity DataIC50: 231nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245645BDBM50245645(CHEMBL4103674)
Affinity DataIC50: 244nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245626BDBM50245626(CHEMBL4094515)
Affinity DataIC50: 273nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase BTK(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245618BDBM50245618(CHEMBL4071893)
Affinity DataIC50: 282nMAssay Description:Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
University of Science and Technology of China

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50245603BDBM50245603(CHEMBL4096207)
Affinity DataIC50: 341nMAssay Description:Inhibition of full length recombinant human N-terminal GST-tagged BMX expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2019
Entry Details Article
PubMed
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