Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50017274
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM35723(N-[4-(7-Chloro-5-hydroxy-2,3,4,5-tetrahydro-benzo[...)
Affinity DataKi:  2.40nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600600(CHEMBL5207885)
Affinity DataKi:  4.30nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600605(CHEMBL5208751)
Affinity DataKi:  9nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600605(CHEMBL5208751)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human V2 receptor expressed in CHO cells assessed as inhibition of vasopressin-induced cAMP accumulation incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600607(CHEMBL5207405)
Affinity DataKi:  10nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600611(CHEMBL5199628)
Affinity DataKi:  12nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600603(CHEMBL5192961)
Affinity DataKi:  12nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600604(CHEMBL5193621)
Affinity DataKi:  13nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600601(CHEMBL5181318)
Affinity DataKi:  18nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600610(CHEMBL5179440)
Affinity DataKi:  23nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600600(CHEMBL5207885)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human V2 receptor expressed in CHO cells assessed as inhibition of vasopressin-induced cAMP accumulation incubated for 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600609(CHEMBL5172250)
Affinity DataKi:  26nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600612(CHEMBL5187046)
Affinity DataKi:  35nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600608(CHEMBL5192496)
Affinity DataKi:  51nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600593(CHEMBL5188374)
Affinity DataKi:  61nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600594(CHEMBL5172734)
Affinity DataKi:  64nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600606(CHEMBL5181341)
Affinity DataKi:  67nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600596(CHEMBL5207214)
Affinity DataKi:  99nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600595(CHEMBL5207597)
Affinity DataKi:  107nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600605(CHEMBL5208751)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]-vasopressin from human V1A receptor expressed in CHO cells membrane by microbeta scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM35723(N-[4-(7-Chloro-5-hydroxy-2,3,4,5-tetrahydro-benzo[...)
Affinity DataKi:  296nMAssay Description:Displacement of [3H]-vasopressin from human V1A receptor expressed in CHO cells membrane by microbeta scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600599(CHEMBL5183482)
Affinity DataKi:  543nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600598(CHEMBL5179419)
Affinity DataKi:  638nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600597(CHEMBL5187312)
Affinity DataKi:  646nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600592(CHEMBL5195053)
Affinity DataKi:  654nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetVasopressin V2 receptor(Human)
Xuzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50600602(CHEMBL5177490)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of conivaptan-red from SNAP-tagged human V2 receptor expressed in HEK293 cells measured after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed