Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50017927
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606242BDBM50606242(CHEMBL5186935)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606235BDBM50606235(CHEMBL5171006)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606253BDBM50606253(CHEMBL5204626)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606234BDBM50606234(CHEMBL5189703)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606238BDBM50606238(CHEMBL5192663)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606239BDBM50606239(CHEMBL5179874)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606233BDBM50606233(CHEMBL5208220)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606237BDBM50606237(CHEMBL5205440)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50308131BDBM50308131(4-{1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]...)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606241BDBM50606241(CHEMBL5196679)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606243BDBM50606243(CHEMBL5204873)
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606245BDBM50606245(CHEMBL5186525)
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human EP4 receptor expressed in CHO cells coexpressing tTA-dependent luciferase reporter and beta arrestin 2-TEV assessed as r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606234BDBM50606234(CHEMBL5189703)
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606236BDBM50606236(CHEMBL5195791)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606247BDBM50606247(CHEMBL5181946)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606251BDBM50606251(CHEMBL5177678)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606245BDBM50606245(CHEMBL5186525)
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606231BDBM50606231(CHEMBL5176688)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606245BDBM50606245(CHEMBL5186525)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human EP4 receptor overexpressed in HEK293 cells assessed as reduction in PGE2-mediated cAMP accumulation preincubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606232BDBM50606232(CHEMBL5202462)
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606240BDBM50606240(CHEMBL5180884)
Affinity DataIC50: 6.60nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119448BDBM119448(US8686018, 107)
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606244BDBM50606244(CHEMBL5202597)
Affinity DataIC50: 9.5nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606218BDBM50606218(CHEMBL5181722)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606229BDBM50606229(CHEMBL5201557)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606222BDBM50606222(CHEMBL5208903)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606227BDBM50606227(CHEMBL5175990)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119448BDBM119448(US8686018, 107)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human EP4 receptor overexpressed in HEK293 cells assessed as reduction in PGE2-mediated cAMP accumulation preincubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606223BDBM50606223(CHEMBL5195058)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606218BDBM50606218(CHEMBL5181722)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606245BDBM50606245(CHEMBL5186525)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606230BDBM50606230(CHEMBL5191478)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606219BDBM50606219(CHEMBL5179032)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606219BDBM50606219(CHEMBL5179032)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606248BDBM50606248(CHEMBL5193793)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606226BDBM50606226(CHEMBL5188328)
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606224BDBM50606224(CHEMBL5203156)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606252BDBM50606252(CHEMBL5196717)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606223BDBM50606223(CHEMBL5195058)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606226BDBM50606226(CHEMBL5188328)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606249BDBM50606249(CHEMBL5190720)
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 119448BDBM119448(US8686018, 107)
Affinity DataIC50: 101nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606250BDBM50606250(CHEMBL5205100)
Affinity DataIC50: 187nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606220BDBM50606220(CHEMBL5181142)
Affinity DataIC50: 206nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606225BDBM50606225(CHEMBL5193807)
Affinity DataIC50: 315nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mouse)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606233BDBM50606233(CHEMBL5208220)
Affinity DataIC50: 336nMAssay Description:Antagonist activity at mouse EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606228BDBM50606228(CHEMBL5199895)
Affinity DataIC50: 642nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606221BDBM50606221(CHEMBL5170985)
Affinity DataIC50: 649nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606246BDBM50606246(CHEMBL5204798)
Affinity DataIC50: 786nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
East China Normal University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50606254BDBM50606254(CHEMBL5194028)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human EP4 receptor transfected in CHO/Galpha16 cells preincubated for 15 mins followed by PGE2 addition by calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
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