Compile Data Set for Download or QSAR
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Found 47 Enz. Inhib. hit(s) with all data for entry = 50019079
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201438((+/-)-5-guanidino-2-(mercaptomethyl)pentanoic acid...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201429(2-(1-carbamimidoylpiperidin-3-yl)-3-mercaptopropan...)
Affinity DataIC50:  3nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201429(2-(1-carbamimidoylpiperidin-3-yl)-3-mercaptopropan...)
Affinity DataIC50:  3nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201427(2-(3-guanidinophenyl)-3-mercaptopropanoic acid | C...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201439(2-(2-chloro-5-guanidinophenyl)-3-mercaptopropanoic...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201427(2-(3-guanidinophenyl)-3-mercaptopropanoic acid | C...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201427(2-(3-guanidinophenyl)-3-mercaptopropanoic acid | C...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201438((+/-)-5-guanidino-2-(mercaptomethyl)pentanoic acid...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201438((+/-)-5-guanidino-2-(mercaptomethyl)pentanoic acid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201439(2-(2-chloro-5-guanidinophenyl)-3-mercaptopropanoic...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201435(2-(mercaptomethyl)-3-(piperidin-4-yl)propanoic aci...)
Affinity DataIC50:  29nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201428(3-mercapto-2-(piperidin-4-yl)propanoic acid | CHEM...)
Affinity DataIC50:  37nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201433(2-(1-carbamimidoylpiperidin-4-yl)-3-mercaptopropan...)
Affinity DataIC50:  45nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201429(2-(1-carbamimidoylpiperidin-3-yl)-3-mercaptopropan...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201429(2-(1-carbamimidoylpiperidin-3-yl)-3-mercaptopropan...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201428(3-mercapto-2-(piperidin-4-yl)propanoic acid | CHEM...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201435(2-(mercaptomethyl)-3-(piperidin-4-yl)propanoic aci...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201437(2-(mercaptomethyl)-3-(piperidin-3-yl)propanoic aci...)
Affinity DataIC50:  129nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201427(2-(3-guanidinophenyl)-3-mercaptopropanoic acid | C...)
Affinity DataIC50:  137nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201427(2-(3-guanidinophenyl)-3-mercaptopropanoic acid | C...)
Affinity DataIC50:  137nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201435(2-(mercaptomethyl)-3-(piperidin-4-yl)propanoic aci...)
Affinity DataIC50:  139nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201429(2-(1-carbamimidoylpiperidin-3-yl)-3-mercaptopropan...)
Affinity DataIC50:  165nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201428(3-mercapto-2-(piperidin-4-yl)propanoic acid | CHEM...)
Affinity DataIC50:  195nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201431(2-(3-aminophenyl)-3-mercaptopropanoic acid | CHEMB...)
Affinity DataIC50:  357nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201437(2-(mercaptomethyl)-3-(piperidin-3-yl)propanoic aci...)
Affinity DataIC50:  420nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201437(2-(mercaptomethyl)-3-(piperidin-3-yl)propanoic aci...)
Affinity DataIC50:  420nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201434(3-mercapto-2-(piperidin-3-yl)propanoic acid | CHEM...)
Affinity DataIC50:  445nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201431(2-(3-aminophenyl)-3-mercaptopropanoic acid | CHEMB...)
Affinity DataIC50:  785nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201430(2-(4-carbamimidoylphenyl)-3-mercaptopropanoic acid...)
Affinity DataIC50:  845nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201430(2-(4-carbamimidoylphenyl)-3-mercaptopropanoic acid...)
Affinity DataIC50:  905nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201430(2-(4-carbamimidoylphenyl)-3-mercaptopropanoic acid...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201432(2-(1-(1-iminoethyl)piperidin-4-yl)-3-mercaptopropa...)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201433(2-(1-carbamimidoylpiperidin-4-yl)-3-mercaptopropan...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201434(3-mercapto-2-(piperidin-3-yl)propanoic acid | CHEM...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201434(3-mercapto-2-(piperidin-3-yl)propanoic acid | CHEM...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201437(2-(mercaptomethyl)-3-(piperidin-3-yl)propanoic aci...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201437(2-(mercaptomethyl)-3-(piperidin-3-yl)propanoic aci...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201433(2-(1-carbamimidoylpiperidin-4-yl)-3-mercaptopropan...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201439(2-(2-chloro-5-guanidinophenyl)-3-mercaptopropanoic...)
Affinity DataIC50:  4.65E+3nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201436(2-(1-(2-aminoacetyl)piperidin-4-yl)-3-mercaptoprop...)
Affinity DataIC50:  4.95E+3nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201432(2-(1-(1-iminoethyl)piperidin-4-yl)-3-mercaptopropa...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201436(2-(1-(2-aminoacetyl)piperidin-4-yl)-3-mercaptoprop...)
Affinity DataIC50:  7.35E+3nMAssay Description:Inhibition of human activated thrombin activatable fibrinolysis inhibitorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase N catalytic chain(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201432(2-(1-(1-iminoethyl)piperidin-4-yl)-3-mercaptopropa...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of human carboxypeptidase NMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201434(3-mercapto-2-(piperidin-3-yl)propanoic acid | CHEM...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201434(3-mercapto-2-(piperidin-3-yl)propanoic acid | CHEM...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201436(2-(1-(2-aminoacetyl)piperidin-4-yl)-3-mercaptoprop...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxypeptidase B(Sus scrofa)
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50201431(2-(3-aminophenyl)-3-mercaptopropanoic acid | CHEMB...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of porcine pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed