Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50029921
LigandPNGBDBM50084848(BIs-cyclo(4N-pentyl-1-(4-methylbenzyl)-4-quinolini...)
Affinity DataIC50:  80nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50289333(21,35-diazonia-2,13-diazaoctacyclo[33.6.2.214,21.1...)
Affinity DataIC50:  90nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50084852(1,14-diazonia-22,33-diazaheptacyclo[32.6.2.214,21....)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50084849(Bis-quinolinium cyclophane analogue | CHEMBL258254...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50084839(Bis-quinolinium cyclophane analogue | CHEMBL6266 |...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50084851(Bis-quinolinium cyclophane analogue | CHEMBL266885...)
Affinity DataIC50:  180nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50054105((Z)-1.1'-[stilbene-4,4'-diylbis(methylene)]bis(4-a...)
Affinity DataIC50:  190nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50054098(1,1'-[biphenyl-3,3'-diylbis(methylene)]-bis(4-amin...)
Affinity DataIC50:  290nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50084846(1-[7-(4-amino-1-quinoliniumylmethyl)-9H-2-fluoreny...)
Affinity DataIC50:  310nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50054103(1,1'-[biphenyl-4,4'-diylbis(methylene)]-bis(4-amin...)
Affinity DataIC50:  380nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50054095(1-{4-[4-(4-amino-1-quinoliniumylmethyl)phenethyl]b...)
Affinity DataIC50:  410nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50054096(1-{4-[4-(4-amino-1-quinoliniumylmethyl)benzyl]benz...)
Affinity DataIC50:  450nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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LigandPNGBDBM50048412(4N-[10-(1-benzyl-4-quinoliniumylamino)decyl]-1-ben...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration of compound required for SKCa blocking action was assessed from its ability to inhibit After hyperpolarisation (AHP) in cult...More data for this Ligand-Target Pair
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