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Found 33 Enz. Inhib. hit(s) with all data for entry = 50029926
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50068362(3-Methoxy-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048233(1-(2-Methoxy-phenyl)-4-(1-phenyl-1H-pyrrol-3-ylmet...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50068364(1-(3-Methoxy-phenyl)-4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50068364(1-(3-Methoxy-phenyl)-4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289383(4-Amino-5-chloro-2-methoxy-N-{2-[4-(2-methoxy-phen...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289385(1-Biphenyl-3-ylmethyl-4-(2-methoxy-phenyl)-piperaz...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289383(4-Amino-5-chloro-2-methoxy-N-{2-[4-(2-methoxy-phen...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50068364(1-(3-Methoxy-phenyl)-4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50052573(5-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289383(4-Amino-5-chloro-2-methoxy-N-{2-[4-(2-methoxy-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289384(8-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50123716(1-(3-Methoxy-phenyl)-5-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50123716(1-(3-Methoxy-phenyl)-5-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289384(8-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50123716(1-(3-Methoxy-phenyl)-5-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(4) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-YM-09151-2 from human Dopamine receptor D4.2 expressed in baculovirus Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50289384(8-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50068362(3-Methoxy-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  141nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052573(5-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052573(5-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50068362(3-Methoxy-N-{2-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50052563(3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-N-(5-metho...)
Affinity DataKi:  253nMAssay Description:Displacement of [3H]-spiperone from Dopamine receptor D2 of rat corpora striata synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article