Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50034734
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280987(1N-[12-isopropyl-2,6-dimethyltricyclo[8.4.0.02,7]t...)
Affinity DataIC50:  1.20E+3nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  1.80E+3nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280987(1N-[12-isopropyl-2,6-dimethyltricyclo[8.4.0.02,7]t...)
Affinity DataIC50:  5.40E+3nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280984(C-((4aS,10aR)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50:  8.00E+3nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280984(C-((4aS,10aR)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50:  2.10E+4nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280986(CHEMBL293419 | N-[3-Acetylamino-3-(4-fluoro-phenyl...)
Affinity DataIC50: >2.50E+4nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280985(2-{[((1R,4aS)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50: >2.50E+4nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280988(CHEMBL542142 | N-tetrahydro-1H-2-pyrrolylmethyl-12...)
Affinity DataIC50:  2.80E+4nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50015214(6-chloro-2-methoxy-9-acridinyl(4-diethylamino-1-me...)
Affinity DataIC50:  3.26E+4nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280985(2-{[((1R,4aS)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50:  3.45E+4nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280988(CHEMBL542142 | N-tetrahydro-1H-2-pyrrolylmethyl-12...)
Affinity DataIC50:  6.20E+4nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280984(C-((4aS,10aR)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50:  7.10E+4nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280986(CHEMBL293419 | N-[3-Acetylamino-3-(4-fluoro-phenyl...)
Affinity DataIC50:  9.05E+4nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50015214(6-chloro-2-methoxy-9-acridinyl(4-diethylamino-1-me...)
Affinity DataIC50:  1.00E+5nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  1.20E+5nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280986(CHEMBL293419 | N-[3-Acetylamino-3-(4-fluoro-phenyl...)
Affinity DataIC50:  1.24E+5nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50015214(6-chloro-2-methoxy-9-acridinyl(4-diethylamino-1-me...)
Affinity DataIC50:  1.30E+5nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280985(2-{[((1R,4aS)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50:  2.20E+5nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50: >2.50E+5nMAssay Description:Tested for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  2.50E+5nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin G/H synthase 1/2(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50280987(1N-[12-isopropyl-2,6-dimethyltricyclo[8.4.0.02,7]t...)
Affinity DataIC50:  3.90E+5nMAssay Description:Tested for its inhibitory activity against PGS (prostaglandin synthetase).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
TBA

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50: >7.50E+5nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In DepthDetails Article