Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50006727
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052734(8-Chloro-3-[(E)-3-(4-dimethylamino-phenyl)-allyl]-...)
Affinity DataKi:  18nMAssay Description:Dopamine receptor D1 antagonistic activity as ability to block dopamine-stimulated adenylate cyclase in rat caudateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50029340(8-Chloro-3-(6-dimethylamino-hexyl)-5-phenyl-2,3,4,...)
Affinity DataKi:  21nMAssay Description:Dopamine receptor D1 antagonistic activity as ability to block dopamine-stimulated adenylate cyclase in rat caudateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50029340(8-Chloro-3-(6-dimethylamino-hexyl)-5-phenyl-2,3,4,...)
Affinity DataKi:  49nMAssay Description:Affinity for Dopamine receptor D1 binding measured by competition against [3H]-SCH- 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052734(8-Chloro-3-[(E)-3-(4-dimethylamino-phenyl)-allyl]-...)
Affinity DataKi:  60.7nMAssay Description:Compound was tested for the Binding affinity against Human cloned Dopamine receptor D1 by Radio ligand ([3H]-SCH-23390) binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052733(8-Chloro-3-[2-(4-dimethylamino-phenyl)-ethyl]-5-ph...)
Affinity DataKi:  88.4nMAssay Description:Affinity for Dopamine receptor D1 binding measured by competition against [3H]-SCH- 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052736(8-Bromo-3-[(E)-3-(4-dimethylamino-phenyl)-allyl]-5...)
Affinity DataKi:  120nMAssay Description:Affinity for dopamine receptor D1 binding measured by competition against [3H]-SCH- 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052732(8-Bromo-5-phenyl-3-((E)-3-phenyl-allyl)-2,3,4,5-te...)
Affinity DataKi:  209nMAssay Description:Affinity for dopamine receptor D1 binding measured by competition against [3H]-SCH- 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052734(8-Chloro-3-[(E)-3-(4-dimethylamino-phenyl)-allyl]-...)
Affinity DataKi:  345nMAssay Description:Affinity for Dopamine receptor D2 binding measured by sulpiride 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50029341(8-Chloro-3-(4-dimethylamino-butyl)-5-phenyl-2,3,4,...)
Affinity DataKi:  811nMAssay Description:Affinity for Dopamine receptor D1 binding measured by competition against [3H]-SCH- 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052736(8-Bromo-3-[(E)-3-(4-dimethylamino-phenyl)-allyl]-5...)
Affinity DataKi:  858nMAssay Description:Affinity for Dopamine receptor D2 binding measured by sulpiride 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052737(CHEMBL423510 | {4-[(E)-3-(7-Chloro-8-methoxy-1-phe...)
Affinity DataKi:  1.72E+3nMAssay Description:Affinity for Dopamine receptor D2 binding measured by sulpiride 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052735(CHEMBL114143 | {4-[(E)-3-(7-Bromo-8-methoxy-1-phen...)
Affinity DataKi:  2.00E+3nMAssay Description:Affinity for Dopamine receptor D2 binding measured by sulpiride 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50029341(8-Chloro-3-(4-dimethylamino-butyl)-5-phenyl-2,3,4,...)
Affinity DataKi:  3.45E+3nMAssay Description:Affinity for Dopamine receptor D2 binding measured by sulpiride 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50029340(8-Chloro-3-(6-dimethylamino-hexyl)-5-phenyl-2,3,4,...)
Affinity DataKi:  4.13E+3nMAssay Description:Affinity for Dopamine receptor D2 binding measured by sulpiride 23390 to rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052737(CHEMBL423510 | {4-[(E)-3-(7-Chloro-8-methoxy-1-phe...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was tested for the Binding affinity against Human cloned Dopamine receptor D1 by Radio ligand ([3H]-SCH-23390) binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50052735(CHEMBL114143 | {4-[(E)-3-(7-Bromo-8-methoxy-1-phen...)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was tested for the Binding affinity against Human cloned Dopamine receptor D1 by Radio ligand ([3H]-SCH-23390) binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed