Compile Data Set for Download or QSAR
maximum 50k data
Found 59 Enz. Inhib. hit(s) with all data for entry = 50003512
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50121710(2-(2,6-Diethyl-phenyl)-4H-isoquinoline-1,3-dione |...)
Affinity DataIC50:  409nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50089194((R)-N*4*-Hydroxy-N*1*-[(S)-1-((S)-2-hydroxymethyl-...)
Affinity DataIC50:  830nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  2.62E+3nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472139(CHEMBL89450)
Affinity DataIC50:  3.17E+3nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472127(CHEMBL315938)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075321(2-(2,6-Diisopropyl-phenyl)-4-hydroxy-isoindole-1,3...)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075333(5-Amino-2-(2,6-diisopropyl-phenyl)-isoindole-1,3-d...)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472138(CHEMBL89868)
Affinity DataIC50:  2.07E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50111210(2-(3,5-Dimethyl-phenyl)-4H-isoquinoline-1,3-dione ...)
Affinity DataIC50:  2.33E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075323(2-(2,6-Diethyl-phenyl)-5-hydroxy-isoindole-1,3-dio...)
Affinity DataIC50:  3.25E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066436(2-(2,6-Dimethyl-phenyl)-5-hydroxy-isoindole-1,3-di...)
Affinity DataIC50:  3.74E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075321(2-(2,6-Diisopropyl-phenyl)-4-hydroxy-isoindole-1,3...)
Affinity DataIC50:  4.32E+4nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075323(2-(2,6-Diethyl-phenyl)-5-hydroxy-isoindole-1,3-dio...)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075328(2-(2,6-Diisopropyl-phenyl)-5-hydroxy-isoindole-1,3...)
Affinity DataIC50:  4.63E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066438(5-Amino-2-(2,6-dimethyl-phenyl)-isoindole-1,3-dion...)
Affinity DataIC50:  5.63E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472133(CHEMBL442758)
Affinity DataIC50:  6.03E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075328(2-(2,6-Diisopropyl-phenyl)-5-hydroxy-isoindole-1,3...)
Affinity DataIC50:  6.49E+4nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472134(CHEMBL87161)
Affinity DataIC50:  6.78E+4nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066436(2-(2,6-Dimethyl-phenyl)-5-hydroxy-isoindole-1,3-di...)
Affinity DataIC50:  7.48E+4nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50050521((2-Dihydroxyborane-pyrrolidin-1-yl)-pyrrolidin-2-y...)
Affinity DataIC50:  8.48E+4nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50066438(5-Amino-2-(2,6-dimethyl-phenyl)-isoindole-1,3-dion...)
Affinity DataIC50:  8.63E+4nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472137(CHEMBL88811)
Affinity DataIC50:  1.12E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472124(CHEMBL89026)
Affinity DataIC50:  1.13E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472126(CHEMBL315662)
Affinity DataIC50:  1.43E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472130(CHEMBL91366)
Affinity DataIC50:  1.58E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472129(CHEMBL89630)
Affinity DataIC50:  1.88E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472132(CHEMBL86373)
Affinity DataIC50:  1.93E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075333(5-Amino-2-(2,6-diisopropyl-phenyl)-isoindole-1,3-d...)
Affinity DataIC50:  2.51E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50089194((R)-N*4*-Hydroxy-N*1*-[(S)-1-((S)-2-hydroxymethyl-...)
Affinity DataIC50: >2.59E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075322(2-(2,6-Dimethyl-phenyl)-4-hydroxy-isoindole-1,3-di...)
Affinity DataIC50:  2.65E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472128(CHEMBL89334)
Affinity DataIC50: >2.79E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075335(2-(2,6-Diisopropyl-phenyl)-5-nitro-isoindole-1,3-d...)
Affinity DataIC50: >2.83E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075331(2-(2,6-Diisopropyl-phenyl)-4-nitro-isoindole-1,3-d...)
Affinity DataIC50: >2.83E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472131(CHEMBL86597)
Affinity DataIC50:  3.04E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472135(CHEMBL88338)
Affinity DataIC50: >3.08E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472135(CHEMBL88338)
Affinity DataIC50: >3.08E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472127(CHEMBL315938)
Affinity DataIC50: >3.11E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50: >3.24E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075329(2-(2,6-Diisopropyl-phenyl)-isoindole-1,3-dione | 2...)
Affinity DataIC50: >3.25E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472126(CHEMBL315662)
Affinity DataIC50: >3.26E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50121710(2-(2,6-Diethyl-phenyl)-4H-isoquinoline-1,3-dione |...)
Affinity DataIC50: >3.40E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472139(CHEMBL89450)
Affinity DataIC50: >3.52E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472136(CHEMBL316290)
Affinity DataIC50: >3.57E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472131(CHEMBL86597)
Affinity DataIC50: >3.57E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472136(CHEMBL316290)
Affinity DataIC50: >3.57E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472132(CHEMBL86373)
Affinity DataIC50: >3.57E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472137(CHEMBL88811)
Affinity DataIC50: >3.74E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075326(4-Amino-2-(2,6-dimethyl-phenyl)-isoindole-1,3-dion...)
Affinity DataIC50: >3.75E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075326(4-Amino-2-(2,6-dimethyl-phenyl)-isoindole-1,3-dion...)
Affinity DataIC50: >3.75E+5nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50472124(CHEMBL89026)
Affinity DataIC50: >3.76E+5nMAssay Description:Inhibitory activity against dipeptidyl peptidase IV (DPP- IV)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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