Compile Data Set for Download or QSAR
Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 10454
TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536418BDBM536418(US11242350, Example 89B:)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536417BDBM536417(US11242350, Example 88)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536420BDBM536420(US11242350, Example 91)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536419BDBM536419(US11242350, Example 90)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536421BDBM536421(US11242350, Example 92)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536330BDBM536330(2-(3',5'-difluoro-2'-isopropyl-4'-((6- (methylsulf...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536333BDBM536333(6-((4'-(1,1,1,3,3,3-hexafluoro-2- hydroxypropan-2-...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536332BDBM536332(2-(2'-ethyl-4'-((4- (methylsulfonyl)piperidin-1- y...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536335BDBM536335(2-(2'-(sec-butyl)-4'-((6- (methylsulfonyl)-2,6- di...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536337BDBM536337(1,1,1,3,3,3-hexafluoro-2-(2'-fluoro- 6'-isopropyl-...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536336BDBM536336(2-(2',3'-difluoro-6'-isopropyl-4'-((6- (methylsulf...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536338BDBM536338(6-((2-ethyl-4'-(1,1,1,3,3,3- hexafluoro-2-hydroxyp...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536342BDBM536342(6-((2-ethyl-4'-(1,1,1,3,3,3- hexafluoro-2-hydroxyp...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536348BDBM536348(2-(2'-(tert-butyl)-4'-((6- (methylsulfonyl)-2,6- d...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536322BDBM536322(US11242350, Example 3)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536321BDBM536321(US11242350, Example 59 | US11242350, Example 56 | ...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536324BDBM536324(US11242350, Example 5)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536323BDBM536323(US11242350, Example 4)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536329BDBM536329(2-(3',6'-difluoro-2'-isopropyl-4'-((6- (methylsulf...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536372BDBM536372(1,1,1,3,3,3 -hexafluoro-2-(2'- isopropyl-4'-((6-(m...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536371BDBM536371(2-(2'-cyclopropyl-4'-((6- (methylsulfonyl)-2,6- di...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536373BDBM536373(1,1,1,3,3,3-hexafluoro-2-(4'-((6- (methylsulfonyl)...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536356BDBM536356(2-(2'-ethyl-4'-((7-(methylsulfonyl)- 2,7-diazaspir...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536355BDBM536355(2-(2'-ethyl-4'-((2-(methylsulfonyl)- 2,6-diazaspir...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536364BDBM536364(2-(2'-ethyl-6'-fluoro-4'-((6- (methylsulfonyl)-2,6...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536363BDBM536363(2-(2'-ethyl-2-fluoro-4'-((6- (methylsulfonyl)-2,6-...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536366BDBM536366(2-(2'-ethyl-3'-fluoro-4'-((6- (methylsulfonyl)-2,6...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536365BDBM536365(2-(2'-ethyl-5'-fluoro-4'-((6- (methylsulfonyl)-2,6...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536368BDBM536368(2-(2'-ethyl-2-methyl-4'-((6- (methylsulfonyl)-2,6-...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536401BDBM536401(US11242350, Example 72)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536404BDBM536404(US11242350, Example 75)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536406BDBM536406(US11242350, Example 77)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536405BDBM536405(US11242350, Example 76)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536408BDBM536408(US11242350, Example 79)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536407BDBM536407(US11242350, Example 78)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536410BDBM536410(US11242350, Example 81)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536409BDBM536409(US11242350, Example 80)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536412BDBM536412(US11242350, Example 83)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536411BDBM536411(US11242350, Example 82)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536414BDBM536414(US11242350, Example 85)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536413BDBM536413(US11242350, Example 84)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536416BDBM536416(US11242350, Example 87)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536415BDBM536415(US11242350, Example 86)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536386BDBM536386(1,1,1,3,3,3-hexafluoro-2-(2'- methoxy-2-methyl-4'-...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536387BDBM536387(7-((2-ethyl-4'-(1,1,1,3,3,3- hexafluoro-2-hydroxyp...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536389BDBM536389(2-(4-(4-ethyl-6-((6-(methylsulfonyl)- 2,6-diazaspi...)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536394BDBM536394(US11242350, Example 65)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536393BDBM536393(US11242350, Example 64)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536398BDBM536398(US11242350, Example 69)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Escalier Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 536397BDBM536397(US11242350, Example 68)
Affinity DataIC50: 50nMAssay Description:Compounds of the present invention were tested in a human RORγ ligand binding assay using a commercially available cell based ligand binding rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2022
Entry Details
US Patent

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