Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 10605
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554135(US11325921, Example 22)
Affinity DataIC50:  6.20nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554134(US11325921, Example 21)
Affinity DataIC50:  8.40nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554136(US11325921, Example 23)
Affinity DataIC50:  11nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554133(US11325921, Example 20)
Affinity DataIC50:  11.4nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554059(US11325921, Example 1)
Affinity DataIC50:  13.3nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554111(US11325921, Example 2 | US11325921, Example 9)
Affinity DataIC50:  17.8nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554139(US11325921, Example 26 | US11325921, Example 27)
Affinity DataIC50:  26nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554116(US11325921, Example 6)
Affinity DataIC50:  27.3nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554111(US11325921, Example 2 | US11325921, Example 9)
Affinity DataIC50:  31.7nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554112(US11325921, Example 3)
Affinity DataIC50:  31.8nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554139(US11325921, Example 26 | US11325921, Example 27)
Affinity DataIC50:  44.7nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554126(US11325921, Example 11)
Affinity DataIC50:  53.9nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554138(US11325921, Example 25)
Affinity DataIC50:  90.2nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554128(US11325921, Example 13)
Affinity DataIC50:  134nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554113(US11325921, Example 4)
Affinity DataIC50:  140nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554120(US11325921, Example 7)
Affinity DataIC50:  248nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554125(US11325921, Example 10)
Affinity DataIC50:  343nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554127(US11325921, Example 12)
Affinity DataIC50:  519nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554121(US11325921, Example 8)
Affinity DataIC50:  635nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-lysine N-methyltransferase 2A/Menin(Homo sapiens (Human))
Sumitomo Dainippon Pharma

US Patent
LigandPNGBDBM554131(US11325921, Example 14)
Affinity DataIC50:  2.40E+3nMAssay Description:Test for Evaluating the Inbinition of the Menin-MLL BindingMenin1-615 wherein 6× His tag and HA tag are inserted in the N-terminus, and myc tag is in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent