Compile Data Set for Download or QSAR
Report error Found 179 Enz. Inhib. hit(s) with all data for entry = 9655
LigandChemical structure of BindingDB Monomer ID 792317BDBM792317(US20260042752, Compound 111 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792357BDBM792357(US20260042752, Compound 151 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792318BDBM792318(US20260042752, Compound 112 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792319BDBM792319(US20260042752, Compound 113 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792316BDBM792316(US20260042752, Compound 110 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792348BDBM792348(3-(5-((3-(2-fluoro-3-(pyridin-4-yl)phenyl)-1,2,4-o...)
Affinity DataEC50: <10nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792350BDBM792350(US20260042752, Compound 144 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792241BDBM792241(3-(5-((3-(2-Fluoro-3-(pyrimidin-4-yl)phenyl)-1,2,4...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792241BDBM792241(3-(5-((3-(2-Fluoro-3-(pyrimidin-4-yl)phenyl)-1,2,4...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792352BDBM792352(US20260042752, Compound 146 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:This cell based assay measures the ability of compounds to inhibit the constitutive cAMP activity of GPR6 receptor expressed in CHO-K1 cells. CHO cel...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792212BDBM792212(US20260042752, Compound 4 | US12565492, Compound 4)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792212BDBM792212(US20260042752, Compound 4 | US12565492, Compound 4)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792213BDBM792213(US20260042752, Compound 5 | US12565492, Compound 5)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792320BDBM792320(US20260042752, Compound 114 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792209BDBM792209(US20260042752, Compound 1 | US12565492, Compound 1)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792326BDBM792326(US20260042752, Compound 120 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792297BDBM792297(US20260042752, Compound 91 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792221BDBM792221(US20260042752, Compound 13 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792222BDBM792222(US20260042752, Compound 14 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792222BDBM792222(US20260042752, Compound 14 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792215BDBM792215(US20260042752, Compound 7 | US12565492, Compound 7)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792216BDBM792216(US20260042752, Compound 8 | US12565492, Compound 8)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792294BDBM792294(US20260042752, Compound 88 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792217BDBM792217(US20260042752, Compound 9 | US12565492, Compound 9)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792218BDBM792218(US20260042752, Compound 10 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792296BDBM792296(US20260042752, Compound 90 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792228BDBM792228(US20260042752, Compound 20 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792305BDBM792305(US20260042752, Compound 99 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792229BDBM792229(US20260042752, Compound 21)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792230BDBM792230(US20260042752, Compound 22 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792331BDBM792331(US20260042752, Compound 125 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792223BDBM792223(US20260042752, Compound 15 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792283BDBM792283(US20260042752, Compound 77 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792223BDBM792223(US20260042752, Compound 15 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792302BDBM792302(US20260042752, Compound 96 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792329BDBM792329(US20260042752, Compound 123 | US12565492, Compound...)
Affinity DataEC50: <10nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792226BDBM792226(US20260042752, Compound 18 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792227BDBM792227(US20260042752, Compound 19 | US12565492, Compound ...)
Affinity DataEC50: <10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792333BDBM792333(US20260042752, Compound 127 | US12565492, Compound...)
Affinity DataEC50:  55nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792334BDBM792334(US20260042752, Compound 128 | US12565492, Compound...)
Affinity DataEC50:  55nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792291BDBM792291(tert-Butyl 4-(3-(5-((3-(2,6-dioxopiperidin-3-yl)-2...)
Affinity DataEC50:  55nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792213BDBM792213(US20260042752, Compound 5 | US12565492, Compound 5)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792214BDBM792214(US20260042752, Compound 6 | US12565492, Compound 6)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792292BDBM792292(4-(3-(5-((3-(2,6-Dioxopiperidin-3-yl)-2-oxo-2,3-di...)
Affinity DataEC50:  55nMAssay Description:HEK293 cell lines stably expressing cloned human NR1/NR2B and NR1/NR2A, respectively, were established according to standard previously described met...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792214BDBM792214(US20260042752, Compound 6 | US12565492, Compound 6)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792335BDBM792335(US20260042752, Compound 129 | US12565492, Compound...)
Affinity DataEC50:  55nMAssay Description:For the detection of SMYD2 cellular methylation activity an In Cell Western (ICW) assay was established. This assay allows rapid processing of multip...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792209BDBM792209(US20260042752, Compound 1 | US12565492, Compound 1)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792210BDBM792210(US20260042752, Compound 2 | US12565492, Compound 2)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792210BDBM792210(US20260042752, Compound 2 | US12565492, Compound 2)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 792219BDBM792219(US20260042752, Compound 11 | US12565492, Compound ...)
Affinity DataEC50:  55nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/24/2026
Entry Details
US Patent

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