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Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 5906
Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99930(US8501729, 25)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99936(US8501729, 32)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99935(US8501729, 31)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334453(CHEMBL1643894 | US8501729, 4 | (S)-5-methyl-2-(qui...)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334445(CHEMBL1643887 | US8501729, 8 | (S)-2-ethyl-7-(quin...)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334442(US8501729, 6 | CHEMBL1643884 | (S)-2-methyl-7-(qui...)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99926(US8501729, 21)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334439(CHEMBL1643883 | US8501729, 12 | (R)-2-methyl-7-(qu...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99932(US8501729, 27)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99931(US8501729, 26)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334448(US8501729, 9 | CHEMBL1641625 | (S)-2-isobutyl-7-(q...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334444(US8501729, 14 | CHEMBL1643886 | (R)-2-ethyl-7-(qui...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334443(US8501729, 13 | CHEMBL1643885 | (R)-4-fluoro-2-met...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99929(US8501729, 24)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334447(CHEMBL1643889 | US8501729, 7 | (S)-2-isopropyl-7-(...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334446(US8501729, 15 | CHEMBL1643888 | (R)-2-isopropyl-7-...)
Affinity DataKi:  3nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99934(US8501729, 29)
Affinity DataKi:  3nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99928(US8501729, 23)
Affinity DataKi:  4nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334441(CHEMBL1643882 | US8501729, 11 | (S)-7-(quinuclidin...)
Affinity DataKi:  5nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334440(US8501729, 16 | CHEMBL1643881 | (R)-7-(quinuclidin...)
Affinity DataKi:  5nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334449(US8501729, 17 | CHEMBL1643890 | (R)-2-benzyl-7-(qu...)
Affinity DataKi:  5nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334451(CHEMBL1643892 | US8501729, 10 | (S)-2-(4-fluorophe...)
Affinity DataKi:  7nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99938(US8501729, 34)
Affinity DataKi:  8nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99939(US8501729, 35)
Affinity DataKi:  13nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99923(US8501729, 5)
Affinity DataKi:  13nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99942(US8501729, 30)
Affinity DataKi:  25nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM50334450(US8501729, 18 | CHEMBL1643891 | (R)-2-(4-fluorophe...)
Affinity DataKi:  29nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99927(US8501729, 22)
Affinity DataKi:  34nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99937(US8501729, 33)
Affinity DataKi:  49nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99925(US8501729, 20)
Affinity DataKi:  57nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99941(US8501729, 38)
Affinity DataKi:  59nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99924(US8501729, 19)
Affinity DataKi:  68nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99933(US8501729, 28)
Affinity DataKi:  108nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent

Target5-hydroxytryptamine receptor 3A(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM99940(US8501729, 37)
Affinity DataKi:  267nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
US Patent