Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 1332
TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312140(US9604931, 15g | 6,8-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  0.480nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312151(US9604931, 15i | (E)-6,8-dihydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  1.66nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312096(US9604931, 12u | 4-bromo-6,8-dihydroxy-2-(4-hydrox...)
Affinity DataKi:  3nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM317457(US9623021, 12z | 4-chloro-6,8-dihydroxy-2-(4-hydro...)
Affinity DataKi:  3nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312149(US9604931, 15h | 6,8-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  3.03nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312139(US9604931, 15c | 2-(3-fluoro-4-hydroxyphenyl)-6,8-...)
Affinity DataKi:  3.96nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312136(US9604931, 14k | 4-bromo-6-hydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  6nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM317459(US9623021, 14m | 6,8-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  7nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312096(US9604931, 12u | 4-bromo-6,8-dihydroxy-2-(4-hydrox...)
Affinity DataKi:  32nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM317457(US9623021, 12z | 4-chloro-6,8-dihydroxy-2-(4-hydro...)
Affinity DataKi:  40nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312134(US9604931, 14I | 4-bromo-6-methoxy-2-(4-methoxyphe...)
Affinity DataKi:  46nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM310198(US9604931, 12b | 4-bromo-6-hydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  49nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312140(US9604931, 15g | 6,8-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  70nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312136(US9604931, 14k | 4-bromo-6-hydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  76nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM317459(US9623021, 14m | 6,8-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  94nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312151(US9604931, 15i | (E)-6,8-dihydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  102nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312149(US9604931, 15h | 6,8-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  124nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM317461(US9623021, 15a | 4-bromo-6-hydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  130nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312139(US9604931, 15c | 2-(3-fluoro-4-hydroxyphenyl)-6,8-...)
Affinity DataKi:  205nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor beta(Human)
Gtx

US Patent
LigandPNGBDBM312137(US9604931, 15a | 6-hydroxy-2-(4-hydroxyphenyl)-4-p...)
Affinity DataKi:  252nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312134(US9604931, 14I | 4-bromo-6-methoxy-2-(4-methoxyphe...)
Affinity DataKi: >394nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM310198(US9604931, 12b | 4-bromo-6-hydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  998nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM317461(US9623021, 15a | 4-bromo-6-hydroxy-2-(4-hydroxyphe...)
Affinity DataKi:  1.78E+3nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent

TargetEstrogen receptor(Human)
Gtx

US Patent
LigandPNGBDBM312137(US9604931, 15a | 6-hydroxy-2-(4-hydroxyphenyl)-4-p...)
Affinity DataKi:  2.10E+3nMAssay Description:Recombinant ER-α or ER-β ligand binding domain (LBD) was combined with [3H]E2 (PerkinElmer, Waltham, Mass.) in buffer A (10 mM Tris, pH 7.4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
US Patent