Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 297
TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263227(US9708370, GHRP-6)
Affinity DataEC50:  3.65nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50: 6.08nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263217(US9708370, DBG-253-10)
Affinity DataEC50:  465nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263226(US9708370, DBG-168-8p)
Affinity DataEC50:  514nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))
Affinity DataIC50: 568nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394997(CHEMBL2163482 | US9708370, DBG-253-6)
Affinity DataEC50:  723nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263218(US9708370, DBG-253-11)
Affinity DataEC50:  729nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394996(CHEMBL2163348 | US9708370, DBG-253-7)
Affinity DataEC50:  771nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)
Affinity DataEC50:  808nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263225(US9708370, DBG-145p)
Affinity DataEC50:  809nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataEC50:  1.20E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394999(CHEMBL2163480 | US9708370, DBG-253-3)
Affinity DataEC50:  1.34E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataIC50: 1.34E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263219(US9708370, DBG-253-12)
Affinity DataEC50:  1.64E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263222(US9708370, DBG-175p)
Affinity DataIC50: 1.80E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataEC50:  2.77E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataIC50: 2.89E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263256(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)
Affinity DataIC50: 2.95E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50: 2.97E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394995(CHEMBL2163483 | US9708370, DBG-253-8)
Affinity DataEC50:  3.25E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50: 3.33E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395019(CHEMBL2163449 | US9708370, CP-2B(v))
Affinity DataIC50: 3.68E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394998(CHEMBL2163481 | US9708370, DBG-253-5)
Affinity DataEC50:  3.74E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM254027(US9708370, DBG-253-4)
Affinity DataEC50:  4.28E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395016(CHEMBL2163452 | US9708370, CP-2B(ii))
Affinity DataIC50: 4.94E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394993(CHEMBL2163485 | US9708370, CP-1A(iv))
Affinity DataIC50: 5.02E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263220(US9708370, DBG-253-13)
Affinity DataEC50:  5.49E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395015(CHEMBL2163453 | US9708370, CP-2B(i))
Affinity DataIC50: 8.17E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263222(US9708370, DBG-175p)
Affinity DataEC50:  8.53E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))
Affinity DataIC50: 8.76E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395015(CHEMBL2163453 | US9708370, CP-2B(i))
Affinity DataIC50: 9.02E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)
Affinity DataIC50: 9.61E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetPlatelet glycoprotein 4(Rat)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395017(CHEMBL2163451 | US9708370, CP-2B(iii))
Affinity DataIC50: 9.66E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395028(CHEMBL2163440 | US9708370, CP-1B(iv))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395026(CHEMBL2163442 | US9708370, CP-1B(ii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395025(CHEMBL2163443 | US9708370, CP-1B(i))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394993(CHEMBL2163485 | US9708370, CP-1A(iv))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263230(US9708370, 41 CP-1A(iii) | US9708370, CP-1A(iii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263241(US9708370, 61 CP-AzaGly-Pro)
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395014(CHEMBL2163454 | US9708370, 60 CP-3(iv))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395013(CHEMBL2163455 | US9708370, 59 CP-3(iii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395019(CHEMBL2163449 | US9708370, CP-2B(v))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395018(CHEMBL2163450 | US9708370, 55 CP-2B(iv))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395017(CHEMBL2163451 | US9708370, CP-2B(iii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395016(CHEMBL2163452 | US9708370, CP-2B(ii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395023(CHEMBL2163445 | US9708370, 50 CP-2A(iv))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395022(CHEMBL2163446 | US9708370, 49 CP-2A(iii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395021(CHEMBL2163447 | US9708370, 48 CP-2A(ii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263244(US9708370, 45 CP-1B(iii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394991(CHEMBL2163438 | US9708370, 40 CP-1A(ii))
Affinity DataIC50: 1.00E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
US Patent

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