Reaction Details Report a problem with these data
Target
Atypical chemokine receptor 3
Ligand
BDBM50250373
Substrate
n/a
Meas. Tech.
ChEMBL_1681650 (CHEMBL4031927)
Ki
34±n/a nM
Citation
Boehm, M; Beaumont, K; Jones, R; Kalgutkar, AS; Zhang, L; Atkinson, K; Bai, G; Brown, JA; Eng, H; Goetz, GH; Holder, BR; Khunte, B; Lazzaro, S; Limberakis, C; Ryu, S; Shapiro, MJ; Tylaska, L; Yan, J; Turner, R; Leung, SSF; Ramaseshan, M; Price, DA; Liras, S; Jacobson, MP; Earp, DJ; Lokey, RS; Mathiowetz, AM; Menhaji-Klotz, E Discovery of Potent and Orally Bioavailable Macrocyclic Peptide-Peptoid Hybrid CXCR7 Modulators. J Med Chem 60:9653-9663 (2017) [PubMed] Article
More Info.:
Target
Name:
Atypical chemokine receptor 3
Synonyms:
ACKR3 | ACKR3_HUMAN | C-X-C chemokine receptor type 7 | C-X-C chemokine receptor type 7 (CXCR7) | CMKOR1 | CXC-R7 | CXCR-7 | CXCR7 | Chemokine orphan receptor 1 | G-protein coupled receptor 159 | G-protein coupled receptor RDC1 homolog | GPR159 | RDC-1 | RDC1
Type:
Enzyme
Mol. Mass.:
41498.84
Organism:
Homo sapiens (Human)
Description:
P25106
Residue:
362
Sequence:
MDLHLFDYSEPGNFSDISWPCNSSDCIVVDTVMCPNMPNKSVLLYTLSFIYIFIFVIGMIANSVVVWVNIQAKTTGYDTHCYILNLAIADLWVVLTIPVWVVSLVQHNQWPMGELTCKVTHLIFSINLFGSIFFLTCMSVDRYLSITYFTNTPSSRKKMVRRVVCILVWLLAFCVSLPDTYYLKTVTSASNNETYCRSFYPEHSIKEWLIGMELVSVVLGFAVPFSIIAVFYFLLARAISASSDQEKHSSRKIIFSYVVVFLVCWLPYHVAVLLDIFSILHYIPFTCRLEHALFTALHVTQCLSLVHCCVNPVLYSFINRNYRYELMKAFIFKYSAKTGLTKLIDASRVSETEYSALEQSTK