Reaction Details Report a problem with these data
Target
Peroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147]
Ligand
BDBM222687
Substrate
n/a
Meas. Tech.
Activation Assay
EC50
1500±n/a nM
Citation
Miura, T; Sato, S; Yamada, H; Tagashira, J; Watanabe, T; Sekimoto, R; Ishida, R; Aoki, H; Ohgiya, T Phenylpyridine derivative and drug containing same US Patent US9315493 Publication Date 4/19/2016
More Info.:
Target
Name:
Peroxisome proliferator-activated receptor gamma [182-505]/Regulatory protein GAL4 [1-147]
Synonyms:
PPARgamma2 - DNA binding domain of Gal4
Type:
DNA-Protein
Mol. Mass.:
n/a
Description:
n/a
Components:
This complex has 2 components.
Component 1
Name:
Regulatory protein GAL4 [1-147]
Synonyms:
DNA-binding transcription factor (GAl4) | GAL4 | GAL4_YEAST
Type:
DNA Binding
Mol. Mass.:
16874.50
Organism:
Saccharomyces bayanus (Yeast)
Description:
amino acids 1 to 147
Residue:
147
Sequence:
MKLLSSIEQACDICRLKKLKCSKEKPKCAKCLKNNWECRYSPKTKRSPLTRAHLTEVESRLERLEQLFLLIFPREDLDMILKMDSLQDIKALLTGLFVQDNVNKDAVTDRLASVETDMPLTLRQHRISATSSSEESSNKGQRQLTVS
Component 2
Name:
Peroxisome proliferator-activated receptor gamma [182-505]
Synonyms:
NR1C3 | PPARG | PPARG_HUMAN | Peroxisome proliferator-activated receptor gamma (PPAR-gamma)
Type:
Protein
Mol. Mass.:
37077.80
Organism:
Human
Description:
amino acids 182 to 505
Residue:
324
Sequence:
IHKKSRNKCQYCRFQKCLAVGMSHNAIRFGRMPQAEKEKLLAEISSDIDQLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY