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Target
Fatty acid-binding protein, liver
Ligand
BDBM8961
Substrate
n/a
Meas. Tech.
ChEMBL_1929092 (CHEMBL4432268)
Kd
900000±n/a nM
Citation
 Hendrick, AG; Müller, I; Willems, H; Leonard, PM; Irving, S; Davenport, R; Ito, T; Reeves, J; Wright, S; Allen, V; Wilkinson, S; Heffron, H; Bazin, R; Turney, J; Mitchell, PJ Identification and Investigation of Novel Binding Fragments in the Fatty Acid Binding Protein 6 (FABP6). J Med Chem 59:8094-102 (2016) [PubMed]  Article 
Target
Name:
Fatty acid-binding protein, liver
Synonyms:
FABP1 | FABPL | FABPL_HUMAN | Fatty acid-binding protein, liver | Liver fatty acid binding protein (human L-FABP T94T)
Type:
Protein
Mol. Mass.:
14208.72
Organism:
Homo sapiens (Human)
Description:
human L-FABP
Residue:
127
Sequence:
MSFSGKYQLQSQENFEAFMKAIGLPEELIQKGKDIKGVSEIVQNGKHFKFTITAGSKVIQNEFTVGEECELETMTGEKVKTVVQLEGDNKLVTTFKNIKSVTELNGDIITNTMTLGDIVFKRISKRI
  
Inhibitor
Name:
BDBM8961
Synonyms:
1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrahydroacridin-9-amine | 9-THA | 9-amino-1,2,3,4-tetrahydroacridine (THA) | CHEMBL1337960 | CHEMBL95 | Cognex | Tacrine | Tracine | US8999994, Tacrine | cid_1935 | tacrine.HCl
Type:
Small organic molecule
Emp. Form.:
C13H14N2
Mol. Mass.:
198.2637
SMILES:
Nc1c2CCCCc2nc2ccccc12
Structure:
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