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Found 3213 with Last Name = 'ito' and Initial = 't'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50325534(CHEMBL267495 | nalfurafine)
Affinity DataKi:  0.0190nMAssay Description:Displacement of [3H]DPDPE from human KOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50596292(CHEMBL5185211)
Affinity DataKi:  0.0272nMAssay Description:Displacement of [3H]DPDPE from human KOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50596293(CHEMBL5188658)
Affinity DataKi:  0.0356nMAssay Description:Displacement of [3H]DPDPE from human KOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185958(CHEMBL205971 | N-(2-methoxybenzyl)-N-(4-chloro-2-p...)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185958(CHEMBL205971 | N-(2-methoxybenzyl)-N-(4-chloro-2-p...)
Affinity DataKi:  0.0740nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122294(CHEMBL292092 | N-(5-fluoro-2-phenoxyphenyl)-N-(2-(...)
Affinity DataKi:  0.0780nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185959(CHEMBL381602 | N-(2-ethoxybenzyl)-N-(4-chloro-2-ph...)
Affinity DataKi:  0.0980nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185959(CHEMBL381602 | N-(2-ethoxybenzyl)-N-(4-chloro-2-ph...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50596292(CHEMBL5185211)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.160nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [11C]DAA1106 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85871(VIP Ala9)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122295(CHEMBL63065 | N-(2-Fluoromethoxy-5-methoxy-benzyl)...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85889(VIP Ala8)
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85873(VIP Ala2)
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185957(CHEMBL205767 | N-(2-isopropoxybenzyl)-N-(4-chloro-...)
Affinity DataKi:  0.190nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85889(VIP Ala8)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Nih

Curated by PDSP Ki Database
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50219966(CHEMBL23959)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85892(VIP Ala28)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85887(VIP Ala11)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50274347((2E)-N-[(5R,6R)-17-(cyclopropylmethyl)-4,5-epoxy-3...)
Affinity DataKi:  0.238nMAssay Description:Displacement of [3H]U69,593 from human kappa opioid receptor expressed in CHO cell membranes by micro-beta scintillation counting methodMore data for this Ligand-Target Pair
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85886(VIP Ala24)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85886(VIP Ala24)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85899(VIP Ala25 | VIP Ala26)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85914(VIP [D- Leu27] | VIP [D-Leu27])
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85871(VIP Ala9)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM85889(VIP Ala8)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM85873(VIP Ala2)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85881(VIP Ala15)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM85871(VIP Ala9)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM85892(VIP Ala28)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85887(VIP Ala11)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)
Affinity DataKi:  0.360nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85909(VIP Ala27)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85878(VIP Ala21)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50219965(CHEMBL430913)
Affinity DataKi:  0.400nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM85886(VIP Ala24)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85887(VIP Ala11)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85873(VIP Ala2)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85914(VIP [D- Leu27] | VIP [D-Leu27])
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM85872(VIP Ala19)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85899(VIP Ala25 | VIP Ala26)
Affinity DataKi:  0.470nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85881(VIP Ala15)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(RAT)
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85871(VIP Ala9)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVIP peptides(Homo sapiens (Human))
National Institutes of Health

Curated by PDSP Ki Database
LigandPNGBDBM85899(VIP Ala25 | VIP Ala26)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rattus norvegicus (rat))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50220479(CHEMBL23342)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Charles River Discovery Research Services

Curated by ChEMBL
LigandPNGBDBM50553757(CHEMBL4746471)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-Ro15-1788 from human GABAA alpha5beta3gamma2 by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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