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Target
Gastrotropin
Ligand
BDBM8961
Substrate
n/a
Meas. Tech.
ChEMBL_1929090 (CHEMBL4432266)
Kd
200000±n/a nM
Citation
 Hendrick, AG; Müller, I; Willems, H; Leonard, PM; Irving, S; Davenport, R; Ito, T; Reeves, J; Wright, S; Allen, V; Wilkinson, S; Heffron, H; Bazin, R; Turney, J; Mitchell, PJ Identification and Investigation of Novel Binding Fragments in the Fatty Acid Binding Protein 6 (FABP6). J Med Chem 59:8094-102 (2016) [PubMed]  Article 
Target
Name:
Gastrotropin
Synonyms:
FABP6 | FABP6_HUMAN | Fatty acid-binding protein 6 | Gastrotropin | I-15P | I-BABP | ILBP | ILLBP
Type:
PROTEIN
Mol. Mass.:
14371.59
Organism:
Homo sapiens
Description:
ChEMBL_118985
Residue:
128
Sequence:
MAFTGKFEMESEKNYDEFMKLLGISSDVIEKARNFKIVTEVQQDGQDFTWSQHYSGGHTMTNKFTVGKESNIQTMGGKTFKATVQMEGGKLVVNFPNYHQTSEIVGDKLVEVSTIGGVTYERVSKRLA
  
Inhibitor
Name:
BDBM8961
Synonyms:
1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrahydroacridin-9-amine | 9-THA | 9-amino-1,2,3,4-tetrahydroacridine (THA) | CHEMBL1337960 | CHEMBL95 | Cognex | Tacrine | Tracine | US8999994, Tacrine | cid_1935 | tacrine.HCl
Type:
Small organic molecule
Emp. Form.:
C13H14N2
Mol. Mass.:
198.2637
SMILES:
Nc1c2CCCCc2nc2ccccc12
Structure:
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