Reaction Details Report a problem with these data
Target
Free fatty acid receptor 1
Ligand
BDBM50392861
Substrate
n/a
Meas. Tech.
ChEMBL_2074517 (CHEMBL4730051)
Kd
5.0±n/a nM
Citation
Furukawa, H; Miyamoto, Y; Hirata, Y; Watanabe, K; Hitomi, Y; Yoshitomi, Y; Aida, J; Noguchi, N; Takakura, N; Takami, K; Miwatashi, S; Hirozane, Y; Hamada, T; Ito, R; Ookawara, M; Moritoh, Y; Watanabe, M; Maekawa, T Design and Identification of a GPR40 Full Agonist ( J Med Chem 63:10352-10379 (2020) [PubMed] Article
More Info.:
Target
Name:
Free fatty acid receptor 1
Synonyms:
FFAR1 | FFAR1_HUMAN | G-protein Coupled Receptor 40 | GPR40
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
31473.32
Organism:
Homo sapiens (Human)
Description:
O14842
Residue:
300
Sequence:
MDLPPQLSFGLYVAAFALGFPLNVLAIRGATAHARLRLTPSLVYALNLGCSDLLLTVSLPLKAVEALASGAWPLPASLCPVFAVAHFFPLYAGGGFLAALSAGRYLGAAFPLGYQAFRRPCYSWGVCAAIWALVLCHLGLVFGLEAPGGWLDHSNTSLGINTPVNGSPVCLEAWDPASAGPARFSLSLLLFFLPLAITAFCYVGCLRALARSGLTHRRKLRAAWVAGGALLTLLLCVGPYNASNVASFLYPNLGGSWRKLGLITGAWSVVLNPLVTGYLGRGPGLKTVCAARTQGGKSQK