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Report error Found 2466 for UniProtKB: P37288
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044777BDBM50044777(CHEBI:34543 | Arginine Vasopressin | Beta-Hypopham...)
Affinity DataEC50:  0.00400nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221813BDBM50221813(HO-LVA | CHEMBL394602)
Affinity DataKi:  0.0320nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 384-well plate membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240628BDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221813BDBM50221813(HO-LVA | CHEMBL394602)
Affinity DataKi:  0.0360nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in CHO cells by polarisation binding assay using 96-well plate membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418929BDBM50418929(CHEMBL1807272)
Affinity DataKi:  0.0372nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418907BDBM50418907(CHEMBL1807267)
Affinity DataKi:  0.0398nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50319772BDBM50319772((2'-methylbiphenyl-4-yl)((1S,5R)-1,3,3-trimethyl-6...)
Affinity DataKi:  0.0500nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50319776BDBM50319776((2,2'-dimethylbiphenyl-4-yl)((1S,5R)-1,3,3-trimeth...)
Affinity DataKi:  0.0600nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 593676BDBM593676(US11578077, Example 71 | 2'-(3-hydroxy-7,7-dimethy...)
Affinity DataKi:  0.0630nMAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2023
Entry Details
US Patent

TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50075724BDBM50075724(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-...)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50075720BDBM50075720((HO-LVA23)2-{2-[3-(4-Hydroxy-phenyl)-2-(methyl-4-H...)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221815BDBM50221815(4-({[(6-{N-[(1S)-5-amino-1-carbamoylpentyl]-1-[(3S...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418909BDBM50418909(CHEMBL1807270)
Affinity DataKi:  0.0955nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641725BDBM50641725(CHEMBL5549819)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50319799BDBM50319799((4-(1H-indol-3-yl)-3-methoxyphenyl)((1S,5R)-1,3,3-...)
Affinity DataKi:  0.100nMAssay Description:Displacement [3H]Arg human recombinant Vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641737BDBM50641737(CHEMBL5565555)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641736BDBM50641736(CHEMBL5573173)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240628BDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human V1a receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282232BDBM50282232(CHEMBL4165132)
Affinity DataEC50:  0.126nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in HEK293 cell membranes assessed as inhibition of AVP-induced increase in Ca2+ flux p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032908BDBM50032908(CHEMBL3342789)
Affinity DataEC50:  0.126nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in HEK293 cell membranes assessed as inhibition of AVP-induced increase in Ca2+ flux p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350874BDBM50350874(CHEMBL1819540)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350866BDBM50350866(CHEMBL1819441)
Affinity DataEC50:  0.155nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50282233BDBM50282233(CHEMBL4173036)
Affinity DataEC50:  0.158nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in HEK293 cell membranes assessed as inhibition of AVP-induced increase in Ca2+ flux p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50032907BDBM50032907(CHEMBL3342790)
Affinity DataEC50:  0.158nMAssay Description:Antagonist activity at human vasopressin 1a receptor expressed in HEK293 cell membranes assessed as inhibition of AVP-induced increase in Ca2+ flux p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50075725BDBM50075725(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(6C-...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50075722BDBM50075722(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(5C-...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240673BDBM50240673(CHEMBL4096848)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50205990BDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human V1A receptor expressed in HEK293 cells assessed as intracellular calcium level measured at 3 secs interval for 5 mins by fu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418906BDBM50418906(CHEMBL1807266)
Affinity DataKi:  0.182nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50114031BDBM50114031(1-[5-Chloro-3-(2-chloro-phenyl)-1-(3,4-dimethoxy-b...)
Affinity DataKi:  0.190nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50205990BDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at recombinant human V1a receptor expressed in HEK293 cells assessed as increase in intracellular calcium level measured at 3 secs i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641712BDBM50641712(CHEMBL5575281)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641727BDBM50641727(CHEMBL5574628)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 593614BDBM593614(5-hydroxy-1'-(4'-oxo-1,3-dihydro-4'H- spiro[indene...)
Affinity DataKi:  0.200nMAssay Description:The human V1a receptor was cloned by RT-PCR from total human liver RNA. The coding sequence was subcloned in an expression vector after sequencing to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2023
Entry Details
US Patent

TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641714BDBM50641714(CHEMBL5569717)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641713BDBM50641713(CHEMBL5563095)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469544BDBM50469544(CHEMBL4281963)
Affinity DataKi:  0.200nMAssay Description:Displacement of [Se-Se]-AVP from human V1A receptor expressed in CHO cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641703BDBM50641703(CHEMBL5575561)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50202918BDBM50202918((S)-N-(2-fluoro-3-(trifluoromethyl)benzyl)-5-(4-cy...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for human cloned vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641730BDBM50641730(CHEMBL5575102)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641722BDBM50641722(CHEMBL5542954)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641721BDBM50641721(CHEMBL5571184)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]vasopressin from human V1A receptor assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418914BDBM50418914(CHEMBL1807281)
Affinity DataKi:  0.209nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418914BDBM50418914(CHEMBL1807281)
Affinity DataKi:  0.209nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350852BDBM50350852(CHEMBL1817706)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221813BDBM50221813(HO-LVA | CHEMBL394602)
Affinity DataKi:  0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 96-well plate membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221813BDBM50221813(HO-LVA | CHEMBL394602)
Affinity DataKi:  0.210nMAssay Description:Inhibition of human vasopressin V1a receptor expressed in COS7 cells by HTRF-FRET assay using 384-well plate membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50075728BDBM50075728(4HOPh(CH2)2CO-DTyr(Me)-Phe-Gln-Asn-Arg-Pro-Lys(6C-...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]- HO-LVA from human Vasopressin V1a receptor in membranes of CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350875BDBM50350875(CHEMBL1819541)
Affinity DataEC50:  0.234nMAssay Description:Agonist activity at recombinant human vasopressin V1a receptor expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Tohoku University and Department of Pharmaceutical Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50418366BDBM50418366(CHEMBL1774023)
Affinity DataKi:  0.234nMAssay Description:Displacement of [3H]AVP from human V1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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