Compile Data Set for Download or QSAR
Report error Found 261 of affinity data for UniProtKB/TrEMBL: Q3SYC2
LigandPNGBDBM50652958(CHEMBL5687004)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50652960(CHEMBL5687021)
Affinity DataIC50: 0.420nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50652959(CHEMBL5687051)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50090510(CHEMBL3581716)
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50617831(CHEMBL5434664)
Affinity DataIC50: 1nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM159725(US9035059, 19-4)
Affinity DataIC50: 2nMAssay Description:A test for MGAT2 inhibitory action of test compounds was conducted in accordance with a partially modified version of the method described in John F....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM50617810(CHEMBL5422037)
Affinity DataIC50: 2nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50617826(CHEMBL5415437)
Affinity DataIC50: 2nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50617828(CHEMBL5424834)
Affinity DataIC50: 2nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50442175(CHEMBL2441597)
Affinity DataIC50: 2nMAssay Description:Inhibition of human MGAT2 by LC/MS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50518069(CHEMBL4542050 | US11479538, Example 22)
Affinity DataIC50: 2nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM50652963(CHEMBL5686988)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM289043(US10093650, Example 20 | US10329273, Example 20 | ...)
Affinity DataIC50: 3nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM50090617(CHEMBL3581734)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50652964(CHEMBL5687022)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50058840(CHEMBL3325734)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human MoGAT-2 expressed in human Caco2 cells assessed as inhibition of 2-O-Hexadecylglycerol hydrolysis pretreated for 30 mins by LC-MS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/2/2016
Entry Details Article
PubMed
LigandPNGBDBM159734(US9035059, 24-1/24-2 | US9035059, 23-1)
Affinity DataIC50: 4nMT: 2°CAssay Description:An MGAT2 inhibition test for test compounds was conducted in accordance with a partially modified version of the method described in John F. Lockwood...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM159724(US9035059, 19-3)
Affinity DataIC50: 4nMAssay Description:A test for MGAT2 inhibitory action of test compounds was conducted in accordance with a partially modified version of the method described in John F....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM50652953(CHEMBL5686997)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM400245(US10329273, Example 16 | US11479538, Example 16)
Affinity DataIC50: 5nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM289003(US10093650, Example 16 | US10093650, Example 14 | ...)
Affinity DataIC50: 5nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM289021(US10093650, Example 17 | BDBM400246)
Affinity DataIC50: 5nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM38176(US10093650, Example 2 | US10329273, Example 2 | US...)
Affinity DataIC50: 5nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM159732(US9035059, 20-4)
Affinity DataIC50: 5nMT: 2°CAssay Description:An MGAT2 inhibition test for test compounds was conducted in accordance with a partially modified version of the method described in John F. Lockwood...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM50617821(CHEMBL5406388)
Affinity DataIC50: 5nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50617820(CHEMBL5411014)
Affinity DataIC50: 5nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50652961(CHEMBL5687019)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM159705(US9035059, 18-7)
Affinity DataIC50: 7nMAssay Description:A test for MGAT2 inhibitory action of test compounds was conducted in accordance with a partially modified version of the method described in John F....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM50442176(CHEMBL2441598)
Affinity DataIC50: 7nMAssay Description:Inhibition of human MGAT2 by LC/MS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50442178(CHEMBL2441600 | US9187424, 124)
Affinity DataIC50: 7nMAssay Description:Inhibition of human MGAT2 by LC/MS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50518060(CHEMBL4455357)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50617825(CHEMBL5435045)
Affinity DataIC50: 8nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM289026(US10093650, Example 18 | US10329273, Example 18 | ...)
Affinity DataIC50: 8nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM50617832(CHEMBL5401316)
Affinity DataIC50: 8nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50442175(CHEMBL2441597)
Affinity DataIC50: 8nMAssay Description:Inhibition of human MGAT2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM50652962(CHEMBL5687034)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of N-terminal FLAG-tagged full-length human MGAT2 expressed in human FreeStyle 293-F cell membrane using 13Cx18oleoyl-CoA and 2-oleoyl-gly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50617830(CHEMBL5413599)
Affinity DataIC50: 9nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM211296(US10093650, Example 11 | US10329273, Example 11 | ...)
Affinity DataIC50: 9nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM50442176(CHEMBL2441598)
Affinity DataIC50: 9nMAssay Description:Inhibition of human MGAT2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
LigandPNGBDBM159711(US9035059, 18-16)
Affinity DataIC50: 10nMAssay Description:A test for MGAT2 inhibitory action of test compounds was conducted in accordance with a partially modified version of the method described in John F....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM289042(US10093650, Example 19 | US10329273, Example 19 | ...)
Affinity DataIC50: 10nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM50617812(CHEMBL5407931)
Affinity DataIC50: 10nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM289044(US10093650, Example 21 | US10329273, Example 21 | ...)
Affinity DataIC50: 10nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
US Patent

LigandPNGBDBM159740(US9035059, 24-11 | US9035059, 24-5/24-6)
Affinity DataIC50: 10nMT: 2°CAssay Description:An MGAT2 inhibition test for test compounds was conducted in accordance with a partially modified version of the method described in John F. Lockwood...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM159736(US9035059, 23-3)
Affinity DataIC50: 13nMT: 2°CAssay Description:An MGAT2 inhibition test for test compounds was conducted in accordance with a partially modified version of the method described in John F. Lockwood...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM159734(US9035059, 24-1/24-2 | US9035059, 23-1)
Affinity DataIC50: 13nMAssay Description:A test for MGAT2 inhibitory action of test compounds was conducted in accordance with a partially modified version of the method described in John F....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM159730(US9035059, 20-2)
Affinity DataIC50: 14nMT: 2°CAssay Description:An MGAT2 inhibition test for test compounds was conducted in accordance with a partially modified version of the method described in John F. Lockwood...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM50617834(CHEMBL5439792)
Affinity DataIC50: 14nMAssay Description:Inhibition of human MGAT2 by LC-MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM159735(US9035059, 23-2)
Affinity DataIC50: 14nMAssay Description:A test for MGAT2 inhibitory action of test compounds was conducted in accordance with a partially modified version of the method described in John F....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2015
Entry Details
US Patent

LigandPNGBDBM50442178(CHEMBL2441600 | US9187424, 124)
Affinity DataIC50: 15nMAssay Description:Inhibition of human MGAT2 by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
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