Compile Data Set for Download or QSAR
maximum 50k data
Found 291 of affinity data for UniProtKB/TrEMBL: O54798
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]Bag-3 from mouse BRS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataIC50:  5.40nMAssay Description:Displacement of [3H]Bag-3 from mouse BRS-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50314969(2-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...)
Affinity DataIC50:  6.90nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from mouse BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  33nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447505(CHEMBL3115391)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447504(CHEMBL3115392)
Affinity DataEC50:  227nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447503(CHEMBL3115393)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447502(CHEMBL3115394)
Affinity DataEC50:  46nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447501(CHEMBL3115395)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447497(CHEMBL3115399)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447492(CHEMBL3115373)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447489(CHEMBL3115376)
Affinity DataEC50:  569nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447488(CHEMBL3115377)
Affinity DataEC50:  52nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447487(CHEMBL3115378)
Affinity DataEC50:  62nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447486(CHEMBL3115379)
Affinity DataEC50:  121nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447480(CHEMBL3115385)
Affinity DataEC50:  15nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447478(CHEMBL3115387)
Affinity DataEC50:  3.12E+3nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447476(CHEMBL3115389)
Affinity DataEC50:  62nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041414(CHEMBL3356402)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041415(CHEMBL3356403)
Affinity DataEC50:  282nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041416(CHEMBL3356404)
Affinity DataEC50:  43nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041417(CHEMBL3356405)
Affinity DataEC50:  35nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041418(CHEMBL3356406)
Affinity DataEC50:  81nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041420(CHEMBL3356407)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041421(CHEMBL3356408)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041422(CHEMBL3356409)
Affinity DataEC50:  45nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041423(CHEMBL3356410)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041424(CHEMBL3356411)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041425(CHEMBL3356412)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50041426(CHEMBL3356413)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50381914(CHEMBL2023109 | MK-7725)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447474(CHEMBL3115370)
Affinity DataEC50:  256nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50447473(CHEMBL3115369)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50313751(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataEC50:  9.60nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316909(5-(4'-(2-(4-(cyclopentylmethyl)-2H-imidazol-2-yl)e...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316910(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316911(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316912(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316913(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316914(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316915(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316904(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316905((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50316906((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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