TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.91E+4nMAssay Description:Agonist activity at recombinant human TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for 5 mins by Fl...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 9.60E+4nMAssay Description:Agonist activity at recombinant human TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ level pre-incubated for 5 mins by Fl...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 6.92E+3nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.49E+5nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 9.00E+3nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 6.10E+4nMAssay Description:Agonist activity at human TRPA1 in WI38 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 3.16E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.58E+5nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 7.94E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.12E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 8.51E+3nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 3.16E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 6.03E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.66E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.82E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 3.55E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 4.57E+8nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.70E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.20E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 7.50E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 4.90E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.70E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 7.00E+3nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.60E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 6.30E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 3.50E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.34E+8nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by calcium-3 dye based FLIPR analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.61E+5nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 assessed as increase in calcium influx by two electrode voltage clamp methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.10E+5nMAssay Description:Agonist activity at human TRPA1 in WI38 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 4.90E+3nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Calcium-5 dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 4.20E+6nMAssay Description:Agonist activity at human TRPA1 expressed in CHO cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.15E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.26E+5nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 1.70E+5nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 2.19E+5nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences
Curated by ChEMBL
Hyogo University of Health Sciences
Curated by ChEMBL
Affinity DataEC50: 4.20E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as increase in calcium influx by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair




































