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TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKd:  2.40nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKd:  15nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKd:  398nMAssay Description:Binding affinity to mouse uPA by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKd:  354nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKd:  42nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKd:  11nMAssay Description:Binding affinity to mouse uPA expressed in HEK2936E cells by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92479(Tannic Acid, A | Tannic acid)
Affinity DataIC50: 4.10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50228412(methyl 1-(bis(4-acetamidophenoxy)phosphoryl)-2-(4g...)
Affinity DataIC50: 8nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92485(CDE-066 | US9120744, CDE-066)
Affinity DataIC50: 10nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 10nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured immediatelyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 11nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 8 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 12nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50228418(methyl 1-(diphenoxyphosphoryl)-2-(4-guanidinopheny...)
Affinity DataIC50: 32nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 71nMAssay Description:Inhibition of uPA in presence of 75% mouse serum measured at 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92486(CDE-082 | US9120744, CDE-082)
Affinity DataIC50: 79nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92487(CDE-031 | US9120744, CDE-031)
Affinity DataIC50: 132nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92482(CDE-008 | US9120744, CDE-008)
Affinity DataIC50: 162nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50467212(CHEMBL4285028)
Affinity DataIC50: 410nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92483(CDE-034 | US9120744, CDE-034)
Affinity DataIC50: 644nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM92484(CDE-056 | US9120744, CDE-056)
Affinity DataIC50: 758nMpH: 7.8 T: 2°CAssay Description:Enzyme activity assay using human and murine PAI-1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2012
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataIC50: 5.02E+3nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50529246(CHEMBL4473654)
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataIC50: 3.94E+4nMAssay Description:Inhibition of the intrinsic peri-cellular uPA in mouse CT26 cells assessed as reduction in cell invasion measured every hour by transwell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKi:  6.80nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)
Affinity DataKi:  15nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  20nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  20nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)
Affinity DataKi:  45nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)
Affinity DataKi:  246nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50529264(CHEMBL4513418)
Affinity DataKi:  956nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)
Affinity DataKi:  1.61E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)
Affinity DataKi:  1.77E+3nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataKi:  2.31E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459080(CHEMBL4211423)
Affinity DataKi:  2.77E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459079(CHEMBL4206764)
Affinity DataKi:  3.29E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM81818(CHEMBL1909810 | NSC_1794 | CAS_1794 | HMA)
Affinity DataKi:  9.31E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499242(CHEMBL3736473)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed