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TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.512nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50305818(cid_45281794 | CHEMBL593506 | 1-(biphenyl-4-ylmeth...)
Affinity DataEC50: >442nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50305819(cid_45281797 | CHEMBL603445 | 1-(4-(thiophen-3-yl)...)
Affinity DataEC50: >442nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  1.71E+3nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  210nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50240694(CHEMBL4067722)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human muscarinic acetylcholine receptor M5 expressed in CHO cells assessed as increase in calcium mobilization incubated for 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50249403(CHEMBL4091821)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at human M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50451883(CHEMBL4211076)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of human M5 receptor assessed as increase in acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50452393(CHEMBL4212760)
Affinity DataEC50:  1.30E+3nMAssay Description:Positive allosteric modulation of M5 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50464171(CHEMBL4238059)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human M5 receptor expressed in CHO cells assessed as increase in acetylcholine-induced calcium mobilization pretrea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475440(CHEMBL193698)
Affinity DataEC50:  4.36E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475441(CHEMBL62560)
Affinity DataEC50:  1.47E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475442(CHEMBL194847)
Affinity DataEC50:  263nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475443(CHEMBL364454)
Affinity DataEC50:  26.9nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475444(CHEMBL196219)
Affinity DataEC50:  1.99E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475445(CHEMBL196238)
Affinity DataEC50:  3.01E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475446(CHEMBL196151)
Affinity DataEC50:  93.3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475447(CHEMBL193642)
Affinity DataEC50:  4.46E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475448(CHEMBL195011)
Affinity DataEC50:  1.74nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475449(CHEMBL197092)
Affinity DataEC50:  79.4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475450(CHEMBL194196)
Affinity DataEC50:  89.1nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475451(CHEMBL195939)
Affinity DataEC50:  4.26E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475452(CHEMBL425911)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50064612(Acetic acid 8-methyl-8-aza-bicyclo[3.2.1]oct-6-yl ...)
Affinity DataEC50:  2.45E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475453(CHEMBL372536)
Affinity DataEC50:  50.1nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475454(CHEMBL196218)
Affinity DataEC50:  4.79nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475455(CHEMBL193968)
Affinity DataEC50:  4.07E+5nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475456(CHEMBL196931)
Affinity DataEC50:  1.17E+5nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50064609(Acetic acid 8-aza-bicyclo[3.2.1]oct-6-yl ester | 6...)
Affinity DataEC50:  6.17nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475457(CHEMBL373341)
Affinity DataEC50:  104nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475458(CHEMBL194793)
Affinity DataEC50:  44.7nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475459(CHEMBL194008)
Affinity DataEC50:  6.46nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475460(CHEMBL193341 | CHEBI:31167)
Affinity DataEC50:  7.94E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475461(CHEMBL194144)
Affinity DataEC50:  1.14E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  1.09E+4nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50385682(CHEMBL390842)
Affinity DataEC50:  3.71E+3nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50003014(CHEMBL228144)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50003014(CHEMBL228144)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035277(3-Prop-2-ynyloxy-5,6,7,8-tetrahydro-4H-isoxazolo[4...)
Affinity DataEC50:  950nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  360nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035279(3-Methoxy-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-c]az...)
Affinity DataEC50:  4.70E+3nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataEC50:  55nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM46858(cid_9301 | ARECOLINE HYDROBROMIDE | SMR000058258 |...)
Affinity DataEC50:  600nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035278(3-Ethoxy-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-c]aze...)
Affinity DataEC50:  2.10E+3nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035280(3-Isopropoxy-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-c...)
Affinity DataEC50:  110nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50023229(CHEMBL3329755)
Affinity DataEC50:  190nMAssay Description:Positive allosteric modulation of M5 AchR (unknown origin) assessed as increase in acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50546065(CHEMBL4795177)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of human M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  8.90E+3nMAssay Description:Agonistic activity against muscarinic acetylcholine receptor M5 expressed in NIH 3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataEC50:  630nMAssay Description:Agonistic activity against muscarinic acetylcholine receptor M5 expressed in NIH 3T3 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50568250(CHEMBL4847801)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of human muscarinic acetylcholine M5 receptor expressed in CHO cells in presence of acetylcholine at EC20 concentratio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
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