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TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353018(CHEMBL1821980 | CHEMBL1852660)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of pig APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353018(CHEMBL1821980 | CHEMBL1852660)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of porcine kidney APN using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataKi:  0.5nMAssay Description:Competitive inhibition of pig APN using L-leucine-p-nitroanilide as substrate by Dixon-plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457465(CHEMBL4204736)
Affinity DataKi:  0.600nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50002035(CHEMBL17107 | (2-Hydroxycarbamoyl-3-phenyl-propion...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457475(CHEMBL4216408)
Affinity DataKi:  1.5nMAssay Description:Inhibition of APN in porcine kidney using Ala-p-NA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50393210(CHEMBL1235787)
Affinity DataKi:  1.5nMAssay Description:Inhibition of porcine APNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025070(CHEMBL3355110)
Affinity DataKi:  1.5nMAssay Description:Inhibition of pig recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087089((2S)-2-[(2S)-3-{[(1S)-1-azaniumyl-2-phenylethyl](h...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087095(1-{[3-(4-Bromo-phenyl)-2-(1-carboxy-ethylcarbamoyl...)
Affinity DataKi:  1.90nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105574(CHEMBL3597443)
Affinity DataKi:  2nMAssay Description:Inhibition of porcine kidney APN assessed as decrease in p-nitroanilide release using L-leucine-p-nitroanilide as substrate by spectrophotometric ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50002022(CHEMBL16779 | (2-Benzyl-3-hydroxycarbamoyl-propion...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087097(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  2.20nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for A+B stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087097(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  2.20nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087084(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  2.30nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50078127(2-{3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoy...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087093(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  2.30nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087094((R,S,S)1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-4...)
Affinity DataKi:  2.30nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025913([2-(Formyl-hydroxy-amino)-3-phenyl-propionylamino]...)
Affinity DataIC50: 2.5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50405292(CHEMBL2079630)
Affinity DataKi:  2.90nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087106((2S)-2-[(2S)-3-{[(1S)-1-azaniumylethyl](hydroxy)ph...)
Affinity DataKi:  2.90nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50078134(2-{3-[(1-Amino-2-phenyl-ethyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  2.90nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for A+B stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087089((2S)-2-[(2S)-3-{[(1S)-1-azaniumyl-2-phenylethyl](h...)
Affinity DataKi:  2.90nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105625(CHEMBL3597456)
Affinity DataKi:  3nMAssay Description:Inhibition of porcine kidney APN assessed as decrease in p-nitroanilide release using L-leucine-p-nitroanilide as substrate by spectrophotometric ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087114(C-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  3.10nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50078131(2-{3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  3.20nMAssay Description:Inhibitory activity was measured on pig kidney Aminopeptidase N (activity for A+B stereoisomer)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087096(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  3.20nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087105(1-{[3-Biphenyl-4-yl-2-(1-carboxy-2-phenyl-ethylcar...)
Affinity DataKi:  3.70nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105264(2-(2-Benzyl-3-hydroxycarbamoyl-propionylamino)-pro...)
Affinity DataKi:  3.80nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50078135(2-{3-[(Amino-phenyl-methyl)-hydroxy-phosphinoyl]-2...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025099(CHEMBL3355111)
Affinity DataKi:  3.90nMAssay Description:Inhibition of pig recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025066(CHEMBL3355109)
Affinity DataKi:  4.20nMAssay Description:Inhibition of pig recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087111((2S)-2-[(2S)-3-{[(S)-azaniumyl(phenyl)methyl](hydr...)
Affinity DataKi:  4.20nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087098((2S)-2-[(2S)-3-{[azaniumyl(phenyl)methyl](hydroxy)...)
Affinity DataKi:  4.20nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087094((R,S,S)1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-4...)
Affinity DataKi:  4.60nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087113((2S)-2-[(2S)-3-{[(S)-azaniumyl(phenyl)methyl](hydr...)
Affinity DataKi:  4.80nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087119(C-{[3-Biphenyl-4-yl-2-(1-carboxy-2-hydroxy-ethylca...)
Affinity DataKi:  4.90nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against rabbit kidney aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087088((2S)-2-[(2S)-3-[(1-azaniumylethyl)(hydroxy)phospho...)
Affinity DataKi:  5.20nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087085((2S)-2-[(2S)-3-{[(1S)-1-azaniumyl-2-phenylethyl](h...)
Affinity DataKi:  5.30nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105723(CHEMBL3597460)
Affinity DataKi:  6nMAssay Description:Inhibition of porcine kidney APN assessed as decrease in p-nitroanilide release using L-leucine-p-nitroanilide as substrate by spectrophotometric ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353019(CHEMBL1821981)
Affinity DataKi:  6nMAssay Description:Inhibition of porcine kidney APN using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105573(CHEMBL3597442)
Affinity DataKi:  6nMAssay Description:Inhibition of porcine kidney APN assessed as decrease in p-nitroanilide release using L-leucine-p-nitroanilide as substrate by spectrophotometric ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087112(1-{[2-(1-Carboxy-2-phenyl-ethylcarbamoyl)-3-phenyl...)
Affinity DataKi:  6.30nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087109(1-{[3-Biphenyl-4-yl-2-(1-carboxy-3-methyl-butylcar...)
Affinity DataKi:  6.30nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50078137(2-{3-[(1-Amino-3-methylsulfanyl-propyl)-hydroxy-ph...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of pig kidney Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50087102(1-{[2-(1-Carboxy-3-methyl-butylcarbamoyl)-3-phenyl...)
Affinity DataKi:  6.40nMAssay Description:Inhibitory activity on aminopeptidase N (APN) using Ala-pNA as substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353016(CHEMBL1821978)
Affinity DataKi:  7nMAssay Description:Inhibition of porcine kidney APN assessed as decrease in p-nitroanilide release using L-leucine-p-nitroanilide as substrate by spectrophotometric ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353016(CHEMBL1821978)
Affinity DataKi:  7nMAssay Description:Inhibition of porcine kidney APN using L-leucine-p-nitroanilide as substrate after 30 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353016(CHEMBL1821978)
Affinity DataKi:  7nMAssay Description:Inhibition of pig APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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