Compile Data Set for Download or QSAR
maximum 50k data
Found 85 for UniProtKB: P22007
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289981(Prenyl pyrophosphate analogue | {[(2E,6E)-8-[(3-be...)
Affinity DataKi:  380nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289982(Prenyl pyrophosphate analogue)
Affinity DataKi:  700nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289979(Prenyl pyrophosphate analogue | {[(2E)-4-[(3-benzo...)
Affinity DataKi:  960nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289978(Prenyl pyrophosphate analogue | {[(2E)-4-[(3-benzo...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50144314((2E,4E,6E,8E)-3,7,11-trimethyldodeca-2,4,6,8,10-pe...)
Affinity DataKi:  8.80E+3nMAssay Description:Dissociation constant against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50080764((S)-2-({5-[(Benzyl-pyridin-3-yl-amino)-methyl]-2'-...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50067563((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50067584((S)-2-{[5-((R)-2-Amino-3-mercapto-propylamino)-bip...)
Affinity DataIC50:  0.780nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50072626((S)-2-[2-({(S)-2-[2-(4-Cyano-benzylsulfanyl)-acety...)
Affinity DataIC50:  5.40nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104054(4-Methylsulfanyl-2-{[5-(5-phenyl-furan-2-ylmethoxy...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104052(2-{2-[(2-{2-[1-(4-Cyano-benzyl)-4,5-dihydro-1H-imi...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104047((E)-N-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenyl]...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103281(1-(3-Benzoyl-4-diphenylacetylamino-phenylcarbamoyl...)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103269(1-{3-Benzoyl-4-[2-(4-bromo-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  76nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103285(1-[3-Benzoyl-4-(2-p-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  77nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103271(1-(3-Benzoyl-4-phenylmethanesulfonylamino-phenylca...)
Affinity DataIC50:  85nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238364(3-(4-(Methoxycarbonyl)phenyl)-4-cyano-5-(isopropyl...)
Affinity DataIC50:  85nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103280(1-(3-Benzoyl-4-p-tolylmethanesulfonylamino-phenylc...)
Affinity DataIC50:  100nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103262(1-{3-Benzoyl-4-[2-(4-chloro-phenyl)-acetylamino]-p...)
Affinity DataIC50:  105nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238353(3-(4-Chlorophenyl)-4-cyano-5-(isopropylthio)thioph...)
Affinity DataIC50:  110nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103274(1-{3-Benzoyl-4-[2-(4-nitro-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  115nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103261(1-{3-Benzoyl-4-[2-(2,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238367(3-(4-Tolyl)-4-cyano-5-(isopropylthio)thiophene-2-c...)
Affinity DataIC50:  190nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238361(3-(4-Methoxyphenyl)-4-cyano-5-(isopropylthio)thiop...)
Affinity DataIC50:  250nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238356(3-(4-Fluorophenyl)-4-cyano-5-(isopropylthio)thioph...)
Affinity DataIC50:  270nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238371(3-(2-Naphthyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50:  320nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103270(1-{3-Benzoyl-4-[2-(2,6-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  340nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238374(3-(3-Thienyl)-4-cyano-5-(isopropylthio)thiophene-2...)
Affinity DataIC50:  350nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103272(1-[3-Benzoyl-4-(2-naphthalen-1-yl-acetylamino)-phe...)
Affinity DataIC50:  380nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104050(5-Phenyl-pentanoic acid [3-benzoyl-4-(2-p-tolyl-ac...)
Affinity DataIC50:  390nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103260(1-[3-Benzoyl-4-(2-o-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103258(1-{3-Benzoyl-4-[2-(2,3-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  420nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104055(CHEMBL276748 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  455nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103277(1-[3-Benzoyl-4-(2-naphthalen-2-yl-acetylamino)-phe...)
Affinity DataIC50:  460nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238357(3-(3-Fluorophenyl)-4-cyano-5-(isopropylthio)thioph...)
Affinity DataIC50:  460nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103284(1-{3-Benzoyl-4-[2-(3,4-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  480nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104048(CHEMBL106900 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  530nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103276(1-{3-Benzoyl-4-[2-(3,5-dichloro-phenyl)-acetylamin...)
Affinity DataIC50:  535nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103259(1-[3-Benzoyl-4-(2-m-tolyl-acetylamino)-phenylcarba...)
Affinity DataIC50:  540nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103268(1-{3-Benzoyl-4-[2-(4-methoxy-phenyl)-acetylamino]-...)
Affinity DataIC50:  545nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103257(1-[3-Benzoyl-4-(4-carboxy-butyrylamino)-phenylcarb...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238359(3-(4-(Trifluoromethyl)phenyl)-4-cyano-5-(isopropyl...)
Affinity DataIC50:  580nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238366(3-Phenyl-4-cyano-5-(isopropylthio)thiophene-2-carb...)
Affinity DataIC50:  610nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238365(3-(3-(Methoxycarbonyl)phenyl)-4-cyano-5-(isopropyl...)
Affinity DataIC50:  620nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM238373(3-(3-Biphenyl)-4-cyano-5-(isopropylthio)thiophene-...)
Affinity DataIC50:  640nMpH: 7.5Assay Description:Assays were realized on 96-well plates, prepared with Biomek NKMC and Biomek 3000 from Beckman Coulter and read on Wallac Victor fluorimeter from Per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103278(1-[3-Benzoyl-4-(2-phenyl-propionylamino)-phenylcar...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103287(1-(3-Benzoyl-4-phenylacetylamino-phenylcarbamoyl)-...)
Affinity DataIC50:  650nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103266(1-[3-Benzoyl-4-(3-carboxy-propionylamino)-phenylca...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50103283(1-{3-Benzoyl-4-[2-(4-trifluoromethyl-phenyl)-acety...)
Affinity DataIC50:  725nMAssay Description:Inhibitory activity against farnesyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50104053(CHEMBL329401 | N-[3-Benzoyl-4-(2-p-tolyl-acetylami...)
Affinity DataIC50:  925nMAssay Description:Inhibitory activity against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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