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Report error Found 134 of affinity data for UniProtKB/TrEMBL: P22411
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437403(CHEMBL2408771)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437403(CHEMBL2408771)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437404(CHEMBL2408655)
Affinity DataIC50: 1nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437404(CHEMBL2408655)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50287059(CHEMBL274249 | CHEMBL1627326 | (S)-1-(2-Amino-3-me...)
Affinity DataKi:  2nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11928((1S,3S,5S)-2-{[(2S,4S)-4-[(3-chloro-4-cyanophenyl)...)
Affinity DataKi:  3.60nM ΔG°:  -47.7kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50145999((1S,5S)-2-(2-Amino-2-cyclopentyl-acetyl)-2-aza-bic...)
Affinity DataKi:  4nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437395(CHEMBL2408638)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146002((S)-2-((S)-2-Amino-3-methyl-3-(S)-methyl-butyryl)-...)
Affinity DataKi:  7nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146015((1S,5S)-2-[2-Amino-2-(1-methyl-cyclopentyl)-acetyl...)
Affinity DataKi:  7nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146009((1S,5S)-2-[2-Amino-2-(1-methyl-cyclohexyl)-acetyl]...)
Affinity DataKi:  8nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50151003(CHEMBL1627303 | CHEMBL363250 | (S)-1-((S)-2-Amino-...)
Affinity DataKi:  8nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437395(CHEMBL2408638)
Affinity DataIC50: 9nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146010((1S,5S)-2-[2-Amino-2-(1-methyl-cyclobutyl)-acetyl]...)
Affinity DataKi:  11nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146007((1R,5S)-3-((S)-2-Amino-3-methyl-butyryl)-3-aza-bic...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50145997((1S,5S)-2-(2-Amino-2-cyclobutyl-acetyl)-2-aza-bicy...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146013((1R,5S)-3-((S)-2-Amino-3,3-dimethyl-butyryl)-3-aza...)
Affinity DataKi:  14nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50145996((1R,5S)-3-((S)-2-Amino-3-methyl-pentanoyl)-3-aza-b...)
Affinity DataKi:  15nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146005((1S,5S)-2-(2-Amino-2-cyclohexyl-acetyl)-2-aza-bicy...)
Affinity DataKi:  15nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437396(CHEMBL2408651)
Affinity DataIC50: 16nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437402(CHEMBL2408774)
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437396(CHEMBL2408651)
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146000((1S,5S)-2-((S)-2-Amino-3-methyl-pentanoyl)-2-aza-b...)
Affinity DataKi:  25nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146004((1R,5R)-2-((S)-2-Amino-3-methyl-butyryl)-2-aza-bic...)
Affinity DataKi:  29nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11920((1S,3S,5S)-2-{[(2S)-3,3-dimethylpyrrolidin-2-yl]ca...)
Affinity DataKi:  37nM ΔG°:  -42.0kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11927(4-chloro-N-[(3S,5S)-5-{[(1S,3S,5S)-3-cyano-2-azabi...)
Affinity DataKi:  39nM ΔG°:  -41.9kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)
Affinity DataIC50: 40nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50206821((R)-3-amino-1-(2-benzoylpiperazin-1-yl)-4-(2,4,5-t...)
Affinity DataKi:  44nMAssay Description:Inhibition of pig kidney DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11917((1S,3S,5S)-2-[(1S,2S,5R)-3-azabicyclo[3.1.0]hexan-...)
Affinity DataKi:  52nM ΔG°:  -41.2kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50206820((R)-3-amino-1-(2-benzoyl-1,2-diazepan-1-yl)-4-(2,4...)
Affinity DataKi:  56.2nMAssay Description:Inhibition of pig kidney DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11925(9H-fluoren-9-ylmethyl N-[(3S,5S)-5-{[(1S,3S,5S)-3-...)
Affinity DataKi:  57nM ΔG°:  -40.9kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437402(CHEMBL2408774)
Affinity DataIC50: 57nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146006((1S,5S)-2-((S)-2-Amino-3-phenyl-propionyl)-2-aza-b...)
Affinity DataKi:  65nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437398(CHEMBL2408646)
Affinity DataIC50: 84nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310584(CHEMBL1078049 | N-(5-Chloro-pyridin-2-yl)-2-(4-{N-...)
Affinity DataIC50: 88nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310577(CHEMBL1079529 | CHEMBL1077867 | (R)-2-(4-(1-(2-(4-...)
Affinity DataIC50: 90nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310577(CHEMBL1079529 | CHEMBL1077867 | (R)-2-(4-(1-(2-(4-...)
Affinity DataIC50: 98nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146001((1S,5S)-2-((S)-1-Amino-pyrrolidine-2-carbonyl)-2-a...)
Affinity DataKi:  107nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310582(CHEMBL1079156 | CHEMBL1079889 | (R)-N-(5-cyanopyri...)
Affinity DataIC50: 110nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310583(CHEMBL1079157 | CHEMBL1079890 | (R)-N-(2-chloropyr...)
Affinity DataIC50: 119nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310584(CHEMBL1078049 | N-(5-Chloro-pyridin-2-yl)-2-(4-{N-...)
Affinity DataIC50: 120nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310583(CHEMBL1079157 | CHEMBL1079890 | (R)-N-(2-chloropyr...)
Affinity DataIC50: 124nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11919((1S,3S,5S)-2-{[(2S,3S)-3-methylpyrrolidin-2-yl]car...)
Affinity DataKi:  126nM ΔG°:  -39.0kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310582(CHEMBL1079156 | CHEMBL1079889 | (R)-N-(5-cyanopyri...)
Affinity DataIC50: 130nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50437401(CHEMBL2408642)
Affinity DataIC50: 130nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50150851(2-((R)-2-Amino-3-methyl-pentanoyl)-3,4-dihydro-2H-...)
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IV of porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM11926(N-[(3S,5S)-5-{[(1S,3S,5S)-3-cyano-2-azabicyclo[3.1...)
Affinity DataKi:  133nM ΔG°:  -38.9kJ/molepH: 7.4 T: 2°CAssay Description:Inhibition of human DPP-IV activity was measured under steady-state conditions by following the absorbance increase at 405 nm upon the substrate clea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50310580((R)-N-(benzo[d]thiazol-2-yl)-2-(4-(1-(2-(4-cyanoth...)
Affinity DataIC50: 134nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Sanofi-Aventis

Curated by ChEMBL
LigandPNGBDBM50146012((1S,5S)-2-((S)-2-Amino-4-methylsulfanyl-butyryl)-2...)
Affinity DataKi:  135nMAssay Description:In vitro inhibition of porcine Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
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