TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Binding affinity to recombinant Leishmania major NMT assessed as inhibition constantMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant Leishmania major NMT using GCGGSKVKPQPPQA[K-Biotin as peptide substrate incubated for 30 mins by scintillation luminescence...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of Leishmania major NMT H398N mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of Leishmania major NMT H398N mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant Leishmania major NMT using GCGGSKVKPQPPQA[K-Biotin as peptide substrate incubated for 30 mins by scintillation luminescence...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Leishmania major N-myristoyltransferase using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Inhibition of Leishmania major NMT L421Q mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of Leishmania major NMT L421Q mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 7.30nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Inhibition of Leishmania major NMT H398N mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 12nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of Leishmania major NMT H398N mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 25nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition of N-terminal TEV cleavage site-fused His6 tagged Leishmania major NMT (11 to 421 residues) expressed in Escherichia coli Rosetta-2 cells ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 26nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 28nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 35nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 35nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of Leishmania major NMT L421Q mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 39nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Inhibition of Leishmania major NMT L421Q mutant expressed in Escherichia coli Rosetta-2 cells using GSNKSKPK as substrate in presence of MyrCoA after...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 44nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 44nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 45nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Leishmania major)
State University of Paraiba
Curated by ChEMBL
State University of Paraiba
Curated by ChEMBL
Affinity DataIC50: 45nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair






3D Structure (crystal)
































