Compile Data Set for Download or QSAR
Report error Found 752 of affinity data for UniProtKB/TrEMBL: Q9UKP6
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(H-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val-OH | D[CFWKYC]V ...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413764(CHEMBL504097)
Affinity DataKi:  0.282nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50244020(4'-[1-({2-[Cyanomethyl-(3,4-dichloro-phenyl)-amino...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human urotensin-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377218(CHEMBL257171)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377220(CHEMBL255509)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50558696(CHEMBL4777970)
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377217(CHEMBL256989)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)
Affinity DataKi:  0.724nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413762(CHEMBL509604)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50558700(CHEMBL4748168)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413766(CHEMBL510618)
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50558696(CHEMBL4777970)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50002726(CHEMBL2371933)
Affinity DataKi:  0.910nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377215(CHEMBL257415)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048700(CHEMBL3315147)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  1.09nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50002718(CHEMBL385281)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM86516(Urotensin II | ETPDCFWKYCV | L-Ala-Gly-L-Thr-L-Ala...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377227(CHEMBL255462)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(H-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val-OH | D[CFWKYC]V ...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50473964(CHEMBL2370836)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50473964(CHEMBL2370836)
Affinity DataKi:  1.30nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50558695(CHEMBL4741230)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50002725(CHEMBL374468)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413763(CHEMBL448403)
Affinity DataKi:  1.66nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50517327(CHEMBL4472928)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50517320(CHEMBL4568153)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-URP or human [125I[-urotensin-2 from human urotensin 2 receptor expressed in HEK293 or CHOK1 cells after 2 hrs by gamma-counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50112107(Glu-Thr-Pro-Asp-Cys-Phe-Trp-Lys-Tyr-Cys | CHEMBL38...)
Affinity DataEC50:  1.80nMAssay Description:Mobilization of intracellular calcium in CHO cells transiently transfected with human Urotensin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50112120(Cys-Phe-Trp-Lys-Tyr-Cys-Val | CHEMBL53181)
Affinity DataEC50:  1.80nMAssay Description:Mobilization of intracellular calcium in CHO cells transiently transfected with human Urotensin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048703(CHEMBL3315150)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2016
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50112109(Ala-Thr-Pro-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val | CHEM...)
Affinity DataEC50:  1.80nMAssay Description:Mobilization of intracellular calcium in CHO cells transiently transfected with human Urotensin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(H-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val-OH | D[CFWKYC]V ...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at urotensin 2 receptor (unknown origin) expressed in HEK293 cells co-expressing Gq-polycistronic BRET biosensor assessed as inducti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50112110(Glu-Thr-Ala-Asp-Cys-Phe-Trp-Lys-Tyr-Cys-Val | CHEM...)
Affinity DataEC50:  1.90nMAssay Description:Mobilization of intracellular calcium in CHO cells transiently transfected with human Urotensin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
University of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50377224(CHEMBL257767)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]hU-2 from human recombinant Urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
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