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TargetHistone deacetylase 5(Human)
Irbm/Merck Research Laboratories

LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2008
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataEC50:  180nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM25150(Belinostat | (2E)-N-hydroxy-3-[3-(phenylsulfamoyl)...)
Affinity DataEC50:  30nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50465051(CHEMBL4285950)
Affinity DataEC50:  350nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479635(CHEMBL480560)
Affinity DataEC50:  420nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479636(CHEMBL474987)
Affinity DataEC50:  360nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479637(CHEMBL520079)
Affinity DataEC50:  330nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479638(CHEMBL473426)
Affinity DataEC50:  280nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479639(CHEMBL515103)
Affinity DataEC50:  150nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479640(CHEMBL475469)
Affinity DataEC50:  150nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479641(CHEMBL482346)
Affinity DataEC50:  150nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479642(CHEMBL454749)
Affinity DataEC50:  100nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479643(CHEMBL475624)
Affinity DataEC50:  82nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479644(CHEMBL455757)
Affinity DataEC50:  79nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479645(CHEMBL514325)
Affinity DataEC50:  59nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479646(CHEMBL473615)
Affinity DataEC50:  47nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479644(CHEMBL455757)
Affinity DataEC50:  79nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479647(CHEMBL515291)
Affinity DataEC50:  26nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479648(CHEMBL472142)
Affinity DataEC50:  6.71E+4nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479649(CHEMBL480378)
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479650(CHEMBL482165)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479651(CHEMBL521243)
Affinity DataEC50:  950nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479652(CHEMBL480561)
Affinity DataEC50:  460nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataEC50:  550nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479653(CHEMBL481898)
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479654(CHEMBL520109)
Affinity DataEC50:  170nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479655(CHEMBL475468)
Affinity DataEC50:  88nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479656(CHEMBL474427)
Affinity DataEC50:  29nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479657(CHEMBL517242)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479658(CHEMBL480562)
Affinity DataEC50:  280nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479659(CHEMBL474428)
Affinity DataEC50:  160nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479660(CHEMBL514179)
Affinity DataEC50:  100nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479661(CHEMBL473616)
Affinity DataEC50:  91nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479662(CHEMBL480931)
Affinity DataEC50:  50nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479663(CHEMBL482345)
Affinity DataEC50:  850nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479664(CHEMBL520443)
Affinity DataEC50:  1.12E+4nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479665(CHEMBL480588)
Affinity DataEC50:  790nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479666(CHEMBL473821)
Affinity DataEC50:  95nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479667(CHEMBL473820)
Affinity DataEC50:  240nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479668(CHEMBL475788)
Affinity DataEC50:  44nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479669(CHEMBL480589)
Affinity DataEC50:  200nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50479670(CHEMBL475631)
Affinity DataEC50:  42nMAssay Description:Inhibition of histone deacetylase in human HeLa cells assessed as induction of histone H3 hyperacetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483539(CHEMBL1688184)
Affinity DataEC50:  30nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483540(CHEMBL1688186)
Affinity DataEC50:  190nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483541(CHEMBL1688187)
Affinity DataEC50:  460nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483542(CHEMBL1688190)
Affinity DataEC50:  390nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483543(CHEMBL1688191)
Affinity DataEC50:  340nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483544(CHEMBL1688192)
Affinity DataEC50:  6.24E+3nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483545(CHEMBL1688194)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50483546(CHEMBL1688195)
Affinity DataEC50:  2.65E+3nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
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