Affinity DataKi: >1nMAssay Description:Binding affinity to bovine beta-casein A1More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to induced myeloid leukemia cell differentiation protein 1 (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2-like protein 10 [11-204](Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to Bcl-b (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
TargetGlutathione S-transferase Mu 1(Mus musculus)
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse GSTM1-1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of FPPS (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of FPPS (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Affinity DataIC50: 4.82E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin) in baculosomes preincubated for 20 mins followed by addition of CYP enzyme-specific substrate and NADP+ and mea...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) in baculosomes preincubated for 20 mins followed by addition of CYP enzyme-specific substrate and NADP+ and mea...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) in baculosomes preincubated for 20 mins followed by addition of CYP enzyme-specific substrate and NADP+ and mea...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin) in baculosomes preincubated for 20 mins followed by addition of CYP enzyme-specific substrate and NADP+ and mea...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) in baculosomes preincubated for 20 mins followed by addition of CYP enzyme-specific substrate and NADP+ and mea...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin) in baculosomes preincubated for 20 mins followed by addition of CYP enzyme-specific substrate and NADP+ and mea...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Psl Research University
Curated by ChEMBL
Psl Research University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: >5.00E+8nMAssay Description:Inhibition of FPPS (unknown origin)More data for this Ligand-Target Pair
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: >5.00E+8nMAssay Description:Inhibition of FPPS (unknown origin)More data for this Ligand-Target Pair
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: >5.00E+8nMAssay Description:Inhibition of FPPS (unknown origin)More data for this Ligand-Target Pair
TargetFarnesyl pyrophosphate synthase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataIC50: >5.00E+8nMAssay Description:Inhibition of FPPS (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 0nMAssay Description:Binding affinity to acetylcholine esterase (unknown origin)More data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Institut De Chimie Des Substances Naturelles
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Inhibition of Akt1 (unknown origin)More data for this Ligand-Target Pair